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A new synthesis of sulfonamides by aminolysis of p-nitrophenylsulfonates yielding potent and selective adenosine A2B receptor antagonists.
Yan L, Bertarelli DC, Hayallah AM, Meyer H, Klotz KN, Müller CE. Yan L, et al. Among authors: klotz kn. J Med Chem. 2006 Jul 13;49(14):4384-91. doi: 10.1021/jm060277v. J Med Chem. 2006. PMID: 16821798
Introduction of alkynyl chains on C-8 of adenosine led to very selective antagonists of the A(3) adenosine receptor.
Volpini R, Costanzi S, Lambertucci C, Vittori S, Klotz K, Lorenzen A, Cristalli G. Volpini R, et al. Among authors: klotz k. Bioorg Med Chem Lett. 2001 Jul 23;11(14):1931-4. doi: 10.1016/s0960-894x(01)00347-x. Bioorg Med Chem Lett. 2001. PMID: 11459663
Synthesis, biological activity, and molecular modeling investigation of new pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as human A(3) adenosine receptor antagonists.
Baraldi PG, Cacciari B, Moro S, Spalluto G, Pastorin G, Da Ros T, Klotz KN, Varani K, Gessi S, Borea PA. Baraldi PG, et al. Among authors: klotz kn. J Med Chem. 2002 Feb 14;45(4):770-80. doi: 10.1021/jm0109614. J Med Chem. 2002. PMID: 11831890
N(6)-alkyl-2-alkynyl derivatives of adenosine as potent and selective agonists at the human adenosine A(3) receptor and a starting point for searching A(2B) ligands.
Volpini R, Costanzi S, Lambertucci C, Taffi S, Vittori S, Klotz KN, Cristalli G. Volpini R, et al. Among authors: klotz kn. J Med Chem. 2002 Jul 18;45(15):3271-9. doi: 10.1021/jm0109762. J Med Chem. 2002. PMID: 12109910
Medicinal chemistry and pharmacology of A2B adenosine receptors.
Volpini R, Costanzi S, Vittori S, Cristalli G, Klotz KN. Volpini R, et al. Among authors: klotz kn. Curr Top Med Chem. 2003;3(4):427-43. doi: 10.2174/1568026033392264. Curr Top Med Chem. 2003. PMID: 12570760
9-Ethyladenine derivatives as adenosine receptor antagonists: 2- and 8-substitution results in distinct selectivities.
Klotz KN, Kachler S, Lambertucci C, Vittori S, Volpini R, Cristalli G. Klotz KN, et al. Naunyn Schmiedebergs Arch Pharmacol. 2003 Jun;367(6):629-34. doi: 10.1007/s00210-003-0749-9. Epub 2003 May 7. Naunyn Schmiedebergs Arch Pharmacol. 2003. PMID: 12734636
Synthesis, biological evaluation, and molecular modeling of ribose-modified adenosine analogues as adenosine receptor agonists.
Cappellacci L, Franchetti P, Pasqualini M, Petrelli R, Vita P, Lavecchia A, Novellino E, Costa B, Martini C, Klotz KN, Grifantini M. Cappellacci L, et al. Among authors: klotz kn. J Med Chem. 2005 Mar 10;48(5):1550-62. doi: 10.1021/jm049408n. J Med Chem. 2005. PMID: 15743197
Synthesis, biological studies and molecular modeling investigation of 1,3-dimethyl-2,4-dioxo-6-methyl-8-(substituted) 1,2,3,4-tetrahydro [1,2,4]-triazolo [3,4-f]-purines as potential adenosine receptor antagonists.
Pastorin G, Bolcato C, Cacciari B, Kachler S, Klotz KN, Montopoli C, Moro S, Spalluto G. Pastorin G, et al. Among authors: klotz kn. Farmaco. 2005 Apr;60(4):299-306. doi: 10.1016/j.farmac.2005.01.008. Farmaco. 2005. PMID: 15848204
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