Knust H - Search Results

1

Biochemical and behavioural characterization of EMPA, a novel high-affinity, selective antagonist for the OX(2) receptor.

Malherbe P, Borroni E, Gobbi L, Knust H, Nettekoven M, Pinard E, Roche O, Rogers-Evans M, Wettstein JG, Moreau JL. Malherbe P, et al. Among authors: knust h. Br J Pharmacol. 2009 Apr;156(8):1326-41. doi: 10.1111/j.1476-5381.2009.00127.x. Br J Pharmacol. 2009. PMID: 19751316 Free PMC article.

2

RO4938581, a novel cognitive enhancer acting at GABAA alpha5 subunit-containing receptors.

Ballard TM, Knoflach F, Prinssen E, Borroni E, Vivian JA, Basile J, Gasser R, Moreau JL, Wettstein JG, Buettelmann B, Knust H, Thomas AW, Trube G, Hernandez MC. Ballard TM, et al. Among authors: knust h. Psychopharmacology (Berl). 2009 Jan;202(1-3):207-23. doi: 10.1007/s00213-008-1357-7. Epub 2008 Oct 21. Psychopharmacology (Berl). 2009. PMID: 18936916

3

Rational design of novel pyrrolidine derivatives as orally active neurokinin-3 receptor antagonists.

Ratni H, Ballard TM, Bissantz C, Hoffmann T, Jablonski P, Knoflach F, Knust H, Malherbe P, Nettekoven M, Patiny-Adam A, Riemer C, Schmitt M, Spooren W. Ratni H, et al. Among authors: knust h. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6735-8. doi: 10.1016/j.bmcl.2010.08.138. Epub 2010 Sep 17. Bioorg Med Chem Lett. 2010. PMID: 20850972

4

Mapping the binding pocket of a novel, high-affinity, slow dissociating tachykinin NK3 receptor antagonist: biochemical and electrophysiological characterization.

Malherbe P, Knoflach F, Marcuz A, Bohnert C, Weber M, Knust H, Ratni H, Spooren W, Ballard TM, Bissantz C. Malherbe P, et al. Among authors: knust h. Neuropharmacology. 2014 Nov;86:259-72. doi: 10.1016/j.neuropharm.2014.07.017. Epub 2014 Aug 5. Neuropharmacology. 2014. PMID: 25107588

5

Identification of Three Novel Radiotracers for Imaging Aggregated Tau in Alzheimer's Disease with Positron Emission Tomography.

Gobbi LC, Knust H, Körner M, Honer M, Czech C, Belli S, Muri D, Edelmann MR, Hartung T, Erbsmehl I, Grall-Ulsemer S, Koblet A, Rueher M, Steiner S, Ravert HT, Mathews WB, Holt DP, Kuwabara H, Valentine H, Dannals RF, Wong DF, Borroni E. Gobbi LC, et al. Among authors: knust h. J Med Chem. 2017 Sep 14;60(17):7350-7370. doi: 10.1021/acs.jmedchem.7b00632. Epub 2017 Jul 12. J Med Chem. 2017. PMID: 28654263

6

Preclinical Evaluation of ¹⁸F-RO6958948, ¹¹C-RO6931643, and ¹¹C-RO6924963 as Novel PET Radiotracers for Imaging Tau Aggregates in Alzheimer Disease.

Honer M, Gobbi L, Knust H, Kuwabara H, Muri D, Koerner M, Valentine H, Dannals RF, Wong DF, Borroni E. Honer M, et al. Among authors: knust h. J Nucl Med. 2018 Apr;59(4):675-681. doi: 10.2967/jnumed.117.196741. Epub 2017 Sep 28. J Nucl Med. 2018. PMID: 28970331 Free PMC article.

7

Adventures in drug-like chemistry space: from oxetanes to spiroazetidines and beyond!

Rogers-Evans M, Knust H, Plancher JM, Carreira EM, Wuitschik G, Burkhard J, Li DB, Guérot C. Rogers-Evans M, et al. Among authors: knust h. Chimia (Aarau). 2014;68(7-8):492-9. doi: 10.2533/chimia.2014.492. Chimia (Aarau). 2014. PMID: 25437389 Free article.

8

Synthesis and structural analysis of a new class of azaspiro[3.3]heptanes as building blocks for medicinal chemistry.

Burkhard JA, Guérot C, Knust H, Rogers-Evans M, Carreira EM. Burkhard JA, et al. Among authors: knust h. Org Lett. 2010 May 7;12(9):1944-7. doi: 10.1021/ol1003302. Org Lett. 2010. PMID: 20356106

9

Synthesis of fluorinated tricyclic scaffolds by intramolecular [2+2] photocycloaddition reactions.

Fort DA, Woltering TJ, Nettekoven M, Knust H, Bach T. Fort DA, et al. Among authors: knust h. Angew Chem Int Ed Engl. 2012 Oct 1;51(40):10169-72. doi: 10.1002/anie.201204080. Epub 2012 Sep 7. Angew Chem Int Ed Engl. 2012. PMID: 22962009 No abstract available.

10

Conformationally restricted pyrrolidines by intramolecular [2+2] photocycloaddition reactions.

Fort DA, Woltering TJ, Nettekoven M, Knust H, Bach T. Fort DA, et al. Among authors: knust h. Chem Commun (Camb). 2013 Apr 14;49(29):2989-91. doi: 10.1039/c3cc40757h. Chem Commun (Camb). 2013. PMID: 23463393

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