Labesse G - Search Results

1

6-(Hetero)Arylpurine nucleotides as inhibitors of the oncogenic target DNPH1: synthesis, structural studies and cytotoxic activities.

Amiable C, Paoletti J, Haouz A, Padilla A, Labesse G, Kaminski PA, Pochet S. Amiable C, et al. Among authors: labesse g. Eur J Med Chem. 2014 Oct 6;85:418-37. doi: 10.1016/j.ejmech.2014.07.110. Epub 2014 Aug 1. Eur J Med Chem. 2014. PMID: 25108359

2

Thymidylate kinase of Mycobacterium tuberculosis: a chimera sharing properties common to eukaryotic and bacterial enzymes.

Munier-Lehmann H, Chaffotte A, Pochet S, Labesse G. Munier-Lehmann H, et al. Among authors: labesse g. Protein Sci. 2001 Jun;10(6):1195-205. doi: 10.1110/ps.45701. Protein Sci. 2001. PMID: 11369858 Free PMC article.

3

Comparative study of purine and pyrimidine nucleoside analogues acting on the thymidylate kinases of Mycobacterium tuberculosis and of humans.

Pochet S, Dugué L, Labesse G, Delepierre M, Munier-Lehmann H. Pochet S, et al. Among authors: labesse g. Chembiochem. 2003 Aug 4;4(8):742-7. doi: 10.1002/cbic.200300608. Chembiochem. 2003. PMID: 12898625

4

Design of Mycobacterium tuberculosis thymidine monophosphate kinase inhibitors.

Munier-Lehmann H, Pochet S, Dugue L, Dutruel O, Labesse G, Douget D. Munier-Lehmann H, et al. Among authors: labesse g. Nucleosides Nucleotides Nucleic Acids. 2003 May-Aug;22(5-8):801-4. doi: 10.1081/NCN-120022638. Nucleosides Nucleotides Nucleic Acids. 2003. PMID: 14565282 No abstract available.

5

LEA3D: a computer-aided ligand design for structure-based drug design.

Douguet D, Munier-Lehmann H, Labesse G, Pochet S. Douguet D, et al. Among authors: labesse g. J Med Chem. 2005 Apr 7;48(7):2457-68. doi: 10.1021/jm0492296. J Med Chem. 2005. PMID: 15801836

6

Nucleoside analogues as inhibitors of thymidylate kinases: possible therapeutic applications.

Pochet S, Dugue L, Douguet D, Labesse G, Munier-Lehmann H. Pochet S, et al. Among authors: labesse g. Chembiochem. 2002 Jan 4;3(1):108-10. doi: 10.1002/1439-7633(20020104)3:1<108::AID-CBIC108>3.0.CO;2-B. Chembiochem. 2002. PMID: 17590962 No abstract available.

7

NAD kinases use substrate-assisted catalysis for specific recognition of NAD.

Poncet-Montange G, Assairi L, Arold S, Pochet S, Labesse G. Poncet-Montange G, et al. Among authors: labesse g. J Biol Chem. 2007 Nov 23;282(47):33925-34. doi: 10.1074/jbc.M701394200. Epub 2007 Aug 8. J Biol Chem. 2007. PMID: 17686780 Free article.

8

Structural characterization of the mammalian deoxynucleotide N-hydrolase Rcl and its stabilizing interactions with two inhibitors.

Yang Y, Padilla A, Zhang C, Labesse G, Kaminski PA. Yang Y, et al. Among authors: labesse g. J Mol Biol. 2009 Dec 4;394(3):435-47. doi: 10.1016/j.jmb.2009.10.004. Epub 2009 Oct 12. J Mol Biol. 2009. PMID: 19822152

9

In-plate protein crystallization, in situ ligand soaking and X-ray diffraction.

le Maire A, Gelin M, Pochet S, Hoh F, Pirocchi M, Guichou JF, Ferrer JL, Labesse G. le Maire A, et al. Among authors: labesse g. Acta Crystallogr D Biol Crystallogr. 2011 Sep;67(Pt 9):747-55. doi: 10.1107/S0907444911023249. Epub 2011 Aug 9. Acta Crystallogr D Biol Crystallogr. 2011. PMID: 21904027

10

Screening and in situ synthesis using crystals of a NAD kinase lead to a potent antistaphylococcal compound.

Gelin M, Poncet-Montange G, Assairi L, Morellato L, Huteau V, Dugué L, Dussurget O, Pochet S, Labesse G. Gelin M, et al. Among authors: labesse g. Structure. 2012 Jun 6;20(6):1107-17. doi: 10.1016/j.str.2012.03.024. Epub 2012 May 17. Structure. 2012. PMID: 22608967 Free article.

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