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Reversible covalent binding of neratinib to human serum albumin in vitro.
Drug Metab Lett. 2010 Dec;4(4):220-7. doi: 10.2174/187231210792928206.
Drug Metab Lett. 2010.
PMID: 20690900
Characterization of HKI-272 covalent binding to human serum albumin.
Wang J, Li-Chan XX, Atherton J, Deng L, Espina R, Yu L, Horwatt P, Ross S, Lockhead S, Ahmad S, Chandrasekaran A, Oganesian A, Scatina J, Mutlib A, Talaat R.
Wang J, et al. Among authors: lockhead s.
Drug Metab Dispos. 2010 Jul;38(7):1083-93. doi: 10.1124/dmd.110.032292. Epub 2010 Apr 16.
Drug Metab Dispos. 2010.
PMID: 20400660
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Metabolic disposition of enciprazine, a non-benzodiazepine anxiolytic drug, in rat, dog and man.
Scatina JA, Lockhead SR, Cayen MN, Sisenwine SF.
Scatina JA, et al. Among authors: lockhead sr.
Xenobiotica. 1991 Dec;21(12):1591-604. doi: 10.3109/00498259109044408.
Xenobiotica. 1991.
PMID: 1686125
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Synthesis and structure-activity relationship of novel 6-aryl-1,4-dihydrobenzo[d][1,3]oxazine-2-thiones as progesterone receptor modulators leading to the potent and selective nonsteroidal progesterone receptor agonist tanaproget.
Fensome A, Bender R, Chopra R, Cohen J, Collins MA, Hudak V, Malakian K, Lockhead S, Olland A, Svenson K, Terefenko EA, Unwalla RJ, Wilhelm JM, Wolfrom S, Zhu Y, Zhang Z, Zhang P, Winneker RC, Wrobel J.
Fensome A, et al. Among authors: lockhead s.
J Med Chem. 2005 Aug 11;48(16):5092-5. doi: 10.1021/jm050358b.
J Med Chem. 2005.
PMID: 16078826
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5-(3-Cyclopentyl-2-thioxo-2,3-dihydro-1H-benzimidazol-5-yl)-1-methyl-1H-pyrrole-2-carbonitrile: A novel, highly potent, selective, and orally active non-steroidal progesterone receptor agonist.
Zhang P, Terefenko E, Kern J, Fensome A, Trybulski E, Unwalla R, Wrobel J, Lockhead S, Zhu Y, Cohen J, Lacava M, Winneker RC, Zhang Z.
Zhang P, et al. Among authors: lockhead s.
Bioorg Med Chem. 2007 Oct 15;15(20):6556-64. doi: 10.1016/j.bmc.2007.07.011. Epub 2007 Jul 26.
Bioorg Med Chem. 2007.
PMID: 17681796
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(1-(4-(Naphthalen-2-yl)pyrimidin-2-yl)piperidin-4-yl)methanamine: a wingless beta-catenin agonist that increases bone formation rate.
Pelletier JC, Lundquist JT 4th, Gilbert AM, Alon N, Bex FJ, Bhat BM, Bursavich MG, Coleburn VE, Felix LA, Green DM, Green P, Hauze DB, Kharode YP, Lam HS, Lockhead SR, Magolda RL, Matteo JJ, Mehlmann JF, Milligan C, Murrills RJ, Pirrello J, Selim S, Sharp MC, Unwalla RJ, Vera MD, Wrobel JE, Yaworsky P, Bodine PV.
Pelletier JC, et al. Among authors: lockhead sr.
J Med Chem. 2009 Nov 26;52(22):6962-5. doi: 10.1021/jm9014197.
J Med Chem. 2009.
PMID: 19856966
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Osteogenic effects of a potent Src-over-Abl-selective kinase inhibitor in the mouse.
Murrills RJ, Fukayama S, Boschelli F, Matteo JJ, Owens J, Golas JM, Patel D, Lane G, Liu YB, Carter L, Jussif J, Spaulding V, Wang YD, Boschelli DH, McKew JC, Li XJ, Lockhead S, Milligan C, Kharode YP, Diesl V, Bai Y, Follettie M, Bex FJ, Komm B, Bodine PV.
Murrills RJ, et al. Among authors: lockhead s.
J Pharmacol Exp Ther. 2012 Mar;340(3):676-87. doi: 10.1124/jpet.111.185793. Epub 2011 Dec 9.
J Pharmacol Exp Ther. 2012.
PMID: 22171089
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The Apparent Requirement for Protein Synthesis during G2 Phase Is due to Checkpoint Activation.
Lockhead S, Moskaleva A, Kamenz J, Chen Y, Kang M, Reddy AR, Santos SDM, Ferrell JE Jr.
Lockhead S, et al.
Cell Rep. 2020 Jul 14;32(2):107901. doi: 10.1016/j.celrep.2020.107901.
Cell Rep. 2020.
PMID: 32668239
Free PMC article.
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