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Synthesis, molecular modeling, and opioid receptor affinity of 9, 10-diazatricyclo[4.2.1.1(2,5)]decanes and 2,7-diazatricyclo[4.4.0. 0(3,8)]decanes structurally related to 3,8-diazabicyclo[3.2. 1]octanes.
Vianello P, Albinati A, Pinna GA, Lavecchia A, Marinelli L, Borea PA, Gessi S, Fadda P, Tronci S, Cignarella G. Vianello P, et al. Among authors: marinelli l. J Med Chem. 2000 Jun 1;43(11):2115-23. doi: 10.1021/jm991140q. J Med Chem. 2000. PMID: 10841790
Urotensin-II receptor ligands. From agonist to antagonist activity.
Grieco P, Carotenuto A, Campiglia P, Marinelli L, Lama T, Patacchini R, Santicioli P, Maggi CA, Rovero P, Novellino E. Grieco P, et al. Among authors: marinelli l. J Med Chem. 2005 Nov 17;48(23):7290-7. doi: 10.1021/jm058043j. J Med Chem. 2005. PMID: 16279788
Ethyl 8-fluoro-6-(3-nitrophenyl)-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate as novel, highly potent, and safe antianxiety agent.
Anzini M, Braile C, Valenti S, Cappelli A, Vomero S, Marinelli L, Limongelli V, Novellino E, Betti L, Giannaccini G, Lucacchini A, Ghelardini C, Norcini M, Makovec F, Giorgi G, Ian Fryer R. Anzini M, et al. Among authors: marinelli l. J Med Chem. 2008 Aug 14;51(15):4730-43. doi: 10.1021/jm8002944. Epub 2008 Jul 19. J Med Chem. 2008. PMID: 18637672
634 results