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Novel tricyclic-alpha-alkyloxyphenylpropionic acids: dual PPARalpha/gamma agonists with hypolipidemic and antidiabetic activity.
Sauerberg P, Pettersson I, Jeppesen L, Bury PS, Mogensen JP, Wassermann K, Brand CL, Sturis J, Wöldike HF, Fleckner J, Andersen AS, Mortensen SB, Svensson LA, Rasmussen HB, Lehmann SV, Polivka Z, Sindelar K, Panajotova V, Ynddal L, Wulff EM. Sauerberg P, et al. Among authors: mogensen jp. J Med Chem. 2002 Feb 14;45(4):789-804. doi: 10.1021/jm010964g. J Med Chem. 2002. PMID: 11831892
Design and synthesis of novel PPARalpha/gamma/delta triple activators using a known PPARalpha/gamma dual activator as structural template.
Mogensen JP, Jeppesen L, Bury PS, Pettersson I, Fleckner J, Nehlin J, Frederiksen KS, Albrektsen T, Din N, Mortensen SB, Svensson LA, Wassermann K, Wulff EM, Ynddal L, Sauerberg P. Mogensen JP, et al. Bioorg Med Chem Lett. 2003 Jan 20;13(2):257-60. doi: 10.1016/s0960-894x(02)00881-8. Bioorg Med Chem Lett. 2003. PMID: 12482434
Large dimeric ligands with favorable pharmacokinetic properties and peroxisome proliferator-activated receptor agonist activity in vitro and in vivo.
Sauerberg P, Bury PS, Mogensen JP, Deussen HJ, Pettersson I, Fleckner J, Nehlin J, Frederiksen KS, Albrektsen T, Din N, Svensson LA, Ynddal L, Wulff EM, Jeppesen L. Sauerberg P, et al. Among authors: mogensen jp. J Med Chem. 2003 Nov 6;46(23):4883-94. doi: 10.1021/jm0309046. J Med Chem. 2003. PMID: 14584939
Structure-activity relationships of dimeric PPAR agonists.
Sauerberg P, Mogensen JP, Jeppesen L, Svensson LA, Fleckner J, Nehlin J, Wulff EM, Pettersson I. Sauerberg P, et al. Among authors: mogensen jp. Bioorg Med Chem Lett. 2005 Mar 1;15(5):1497-500. doi: 10.1016/j.bmcl.2004.12.084. Bioorg Med Chem Lett. 2005. PMID: 15713415
Identification and synthesis of a novel selective partial PPARdelta agonist with full efficacy on lipid metabolism in vitro and in vivo.
Sauerberg P, Olsen GS, Jeppesen L, Mogensen JP, Pettersson I, Jeppesen CB, Daugaard JR, Galsgaard ED, Ynddal L, Fleckner J, Panajotova V, Polivka Z, Pihera P, Havranek M, Wulff EM. Sauerberg P, et al. Among authors: mogensen jp. J Med Chem. 2007 Apr 5;50(7):1495-503. doi: 10.1021/jm061202u. Epub 2007 Mar 8. J Med Chem. 2007. PMID: 17343371
Design of potent PPARalpha agonists.
Sauerberg P, Mogensen JP, Jeppesen L, Bury PS, Fleckner J, Olsen GS, Jeppesen CB, Wulff EM, Pihera P, Havranek M, Polivka Z, Pettersson I. Sauerberg P, et al. Among authors: mogensen jp. Bioorg Med Chem Lett. 2007 Jun 1;17(11):3198-202. doi: 10.1016/j.bmcl.2007.03.015. Epub 2007 Mar 12. Bioorg Med Chem Lett. 2007. PMID: 17379517
6-Chloro-3-alkylamino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-dioxide derivatives potently and selectively activate ATP sensitive potassium channels of pancreatic beta-cells.
Nielsen FE, Bodvarsdottir TB, Worsaae A, MacKay P, Stidsen CE, Boonen HC, Pridal L, Arkhammar PO, Wahl P, Ynddal L, Junager F, Dragsted N, Tagmose TM, Mogensen JP, Koch A, Treppendahl SP, Hansen JB. Nielsen FE, et al. Among authors: mogensen jp. J Med Chem. 2002 Sep 12;45(19):4171-87. doi: 10.1021/jm0208121. J Med Chem. 2002. PMID: 12213059
Selective PPAR agonists for the treatment of type 2 diabetes.
Nehlin JO, Mogensen JP, Petterson I, Jeppesen L, Fleckner J, Wulff EM, Sauerberg P. Nehlin JO, et al. Among authors: mogensen jp. Ann N Y Acad Sci. 2006 May;1067:448-53. doi: 10.1196/annals.1354.064. Ann N Y Acad Sci. 2006. PMID: 16804025 Review.
15 results