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Targeting Her2-insYVMA with Covalent Inhibitors-A Focused Compound Screening and Structure-Based Design Approach.
J Med Chem. 2020 Oct 22;63(20):11725-11755. doi: 10.1021/acs.jmedchem.0c00870. Epub 2020 Sep 30.
J Med Chem. 2020.
PMID: 32931277
Structure Defines Function: Clinically Relevant Mutations in ErbB Kinases.
Niggenaber J, Hardick J, Lategahn J, Rauh D.
Niggenaber J, et al.
J Med Chem. 2020 Jan 9;63(1):40-51. doi: 10.1021/acs.jmedchem.9b00964. Epub 2019 Aug 28.
J Med Chem. 2020.
PMID: 31414802
Review.
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Inhibition of osimertinib-resistant epidermal growth factor receptor EGFR-T790M/C797S.
Lategahn J, Keul M, Klövekorn P, Tumbrink HL, Niggenaber J, Müller MP, Hodson L, Flaßhoff M, Hardick J, Grabe T, Engel J, Schultz-Fademrecht C, Baumann M, Ketzer J, Mühlenberg T, Hiller W, Günther G, Unger A, Müller H, Heimsoeth A, Golz C, Blank-Landeshammer B, Kollipara L, Zahedi RP, Strohmann C, Hengstler JG, van Otterlo WAL, Bauer S, Rauh D.
Lategahn J, et al. Among authors: niggenaber j.
Chem Sci. 2019 Oct 4;10(46):10789-10801. doi: 10.1039/c9sc03445e. eCollection 2019 Dec 14.
Chem Sci. 2019.
PMID: 31857889
Free PMC article.
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Complex Crystal Structures of EGFR with Third-Generation Kinase Inhibitors and Simultaneously Bound Allosteric Ligands.
Niggenaber J, Heyden L, Grabe T, Müller MP, Lategahn J, Rauh D.
Niggenaber J, et al.
ACS Med Chem Lett. 2020 Nov 5;11(12):2484-2490. doi: 10.1021/acsmedchemlett.0c00472. eCollection 2020 Dec 10.
ACS Med Chem Lett. 2020.
PMID: 33335671
Free PMC article.
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Insight into Targeting Exon20 Insertion Mutations of the Epidermal Growth Factor Receptor with Wild Type-Sparing Inhibitors.
Lategahn J, Tumbrink HL, Schultz-Fademrecht C, Heimsoeth A, Werr L, Niggenaber J, Keul M, Parmaksiz F, Baumann M, Menninger S, Zent E, Landel I, Weisner J, Jeyakumar K, Heyden L, Russ N, Müller F, Lorenz C, Brägelmann J, Spille I, Grabe T, Müller MP, Heuckmann JM, Klebl BM, Nussbaumer P, Sos ML, Rauh D.
Lategahn J, et al. Among authors: niggenaber j.
J Med Chem. 2022 May 12;65(9):6643-6655. doi: 10.1021/acs.jmedchem.1c02080. Epub 2022 Apr 29.
J Med Chem. 2022.
PMID: 35486541
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Addressing the Osimertinib Resistance Mutation EGFR-L858R/C797S with Reversible Aminopyrimidines.
Grabe T, Jeyakumar K, Niggenaber J, Schulz T, Koska S, Kleinbölting S, Beck ME, Müller MP, Rauh D.
Grabe T, et al. Among authors: niggenaber j.
ACS Med Chem Lett. 2023 Apr 18;14(5):591-598. doi: 10.1021/acsmedchemlett.2c00514. eCollection 2023 May 11.
ACS Med Chem Lett. 2023.
PMID: 37197473
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Avapritinib-based SAR studies unveil a binding pocket in KIT and PDGFRA.
Teuber A, Schulz T, Fletcher BS, Gontla R, Mühlenberg T, Zischinsky ML, Niggenaber J, Weisner J, Kleinbölting SB, Lategahn J, Sievers S, Müller MP, Bauer S, Rauh D.
Teuber A, et al. Among authors: niggenaber j.
Nat Commun. 2024 Jan 2;15(1):63. doi: 10.1038/s41467-023-44376-8.
Nat Commun. 2024.
PMID: 38167404
Free PMC article.
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