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5'-C-Ethyl-tetrazolyl-N(6)-substituted adenosine and 2-chloro-adenosine derivatives as highly potent dual acting A1 adenosine receptor agonists and A3 adenosine receptor antagonists.
Petrelli R, Torquati I, Kachler S, Luongo L, Maione S, Franchetti P, Grifantini M, Novellino E, Lavecchia A, Klotz KN, Cappellacci L. Petrelli R, et al. Among authors: Novellino E. J Med Chem. 2015 Mar 12;58(5):2560-6. doi: 10.1021/acs.jmedchem.5b00074. Epub 2015 Feb 27. J Med Chem. 2015. PMID: 25699637
A concerted study using binding measurements, X-ray structural data, and molecular modeling on the stereochemical features responsible for the affinity of 6-arylpyrrolo[2,1-d][1,5]benzothiazepines toward mitochondrial benzodiazepine receptors.
Dalpiaz A, Bertolasi V, Borea PA, Nacci V, Fiorini I, Campiani G, Mennini T, Manzoni C, Novellino E, Greco G. Dalpiaz A, et al. Among authors: Novellino E. J Med Chem. 1995 Nov 10;38(23):4730-8. doi: 10.1021/jm00023a013. J Med Chem. 1995. PMID: 7473601
Novel ligands specific for mitochondrial benzodiazepine receptors: 6-arylpyrrolo[2,1-d][1,5]benzothiazepine derivatives. Synthesis, structure-activity relationships, and molecular modeling studies.
Fiorini I, Nacci V, Ciani SM, Garofalo A, Campiani G, Savini L, Novellino E, Greco G, Bernasconi P, Mennini T. Fiorini I, et al. Among authors: Novellino E. J Med Chem. 1994 May 13;37(10):1427-38. doi: 10.1021/jm00036a007. J Med Chem. 1994. PMID: 8182701
Synthesis, biological activity, and SARs of pyrrolobenzoxazepine derivatives, a new class of specific "peripheral-type" benzodiazepine receptor ligands.
Campiani G, Nacci V, Fiorini I, De Filippis MP, Garofalo A, Ciani SM, Greco G, Novellino E, Williams DC, Zisterer DM, Woods MJ, Mihai C, Manzoni C, Mennini T. Campiani G, et al. Among authors: Novellino E. J Med Chem. 1996 Aug 30;39(18):3435-50. doi: 10.1021/jm960251b. J Med Chem. 1996. PMID: 8784441
Synthesis, structure-activity relationships, and molecular modeling studies of N-(indol-3-ylglyoxylyl)benzylamine derivatives acting at the benzodiazepine receptor.
Da Settimo A, Primofiore G, Da Settimo F, Marini AM, Novellino E, Greco G, Martini C, Giannaccini G, Lucacchini A. Da Settimo A, et al. Among authors: Novellino E. J Med Chem. 1996 Dec 20;39(26):5083-91. doi: 10.1021/jm960240i. J Med Chem. 1996. PMID: 8978839
N'-Phenylindol-3-ylglyoxylohydrazide derivatives: synthesis, structure-activity relationships, molecular modeling studies, and pharmacological action on brain benzodiazepine receptors.
Da Settimo A, Primofiore G, Da Settimo F, Marini AM, Novellino E, Greco G, Gesi M, Martini C, Giannaccini G, Lucacchini A. Da Settimo A, et al. Among authors: Novellino E. J Med Chem. 1998 Sep 24;41(20):3821-30. doi: 10.1021/jm9800301. J Med Chem. 1998. PMID: 9748357
Geometrically and conformationally restrained cinnamoyl compounds as inhibitors of HIV-1 integrase: synthesis, biological evaluation, and molecular modeling.
Artico M, Di Santo R, Costi R, Novellino E, Greco G, Massa S, Tramontano E, Marongiu ME, De Montis A, La Colla P. Artico M, et al. Among authors: Novellino E. J Med Chem. 1998 Oct 8;41(21):3948-60. doi: 10.1021/jm9707232. J Med Chem. 1998. PMID: 9767632
Certain inhibitors, lacking one of the two pharmacophoric catechol hydroxyls, retain moderate potency thanks to nonpharmacophoric fragments (i.e., a m-methoxy group in curcumin) which favorably interact with an "accessory" region of IN. ...
Certain inhibitors, lacking one of the two pharmacophoric catechol hydroxyls, retain moderate potency thanks to nonpharmacophoric fragments …
5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3, 4-dihydropyrimidin-4(3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives.
Mai A, Artico M, Sbardella G, Massa S, Novellino E, Greco G, Loi AG, Tramontano E, Marongiu ME, La Colla P. Mai A, et al. Among authors: Novellino E. J Med Chem. 1999 Feb 25;42(4):619-27. doi: 10.1021/jm980260f. J Med Chem. 1999. PMID: 10052969
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