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Design and Activity of Specific Hypoxia-Inducible Factor-2α (HIF-2α) Inhibitors for the Treatment of Clear Cell Renal Cell Carcinoma: Discovery of Clinical Candidate ( S)-3-((2,2-Difluoro-1-hydroxy-7-(methylsulfonyl)-2,3-dihydro-1 H-inden-4-yl)oxy)-5-fluorobenzonitrile (PT2385).
J Med Chem. 2018 Nov 8;61(21):9691-9721. doi: 10.1021/acs.jmedchem.8b01196. Epub 2018 Oct 18.
J Med Chem. 2018.
PMID: 30289716
A Small-Molecule Antagonist of HIF2α Is Efficacious in Preclinical Models of Renal Cell Carcinoma.
Wallace EM, Rizzi JP, Han G, Wehn PM, Cao Z, Du X, Cheng T, Czerwinski RM, Dixon DD, Goggin BS, Grina JA, Halfmann MM, Maddie MA, Olive SR, Schlachter ST, Tan H, Wang B, Wang K, Xie S, Xu R, Yang H, Josey JA.
Wallace EM, et al. Among authors: olive sr.
Cancer Res. 2016 Sep 15;76(18):5491-500. doi: 10.1158/0008-5472.CAN-16-0473. Epub 2016 Sep 6.
Cancer Res. 2016.
PMID: 27635045
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Comparison of PY 108-068, a new calcium antagonist, with nifedipine in exercise-induced asthma.
Olive SR, Hansen JE, Sue DY, Ben-Dov I, Wasserman K.
Olive SR, et al.
Chest. 1986 Aug;90(2):208-11. doi: 10.1378/chest.90.2.208.
Chest. 1986.
PMID: 3525023
Clinical Trial.
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A case of AIDS in New Orleans.
Olive SR.
Olive SR.
J La State Med Soc. 1983 Sep;135(9):4-5, 7.
J La State Med Soc. 1983.
PMID: 6556216
No abstract available.
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