Oueslati N - Search Results

1

Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites.

Selvam C, Lemasson IA, Brabet I, Oueslati N, Karaman B, Cabaye A, Tora AS, Commare B, Courtiol T, Cesarini S, McCort-Tranchepain I, Rigault D, Mony L, Bessiron T, McLean H, Leroux FR, Colobert F, Daniel H, Goupil-Lamy A, Bertrand HO, Goudet C, Pin JP, Acher FC. Selvam C, et al. Among authors: oueslati n. J Med Chem. 2018 Mar 8;61(5):1969-1989. doi: 10.1021/acs.jmedchem.7b01438. Epub 2018 Feb 14. J Med Chem. 2018. PMID: 29397723

2

Synthesis and biological evaluation of 1-amino-2-phosphonomethylcyclopropanecarboxylic acids, new group III metabotropic glutamate receptor agonists.

Sibille P, Lopez S, Brabet I, Valenti O, Oueslati N, Gaven F, Goudet C, Bertrand HO, Neyton J, Marino MJ, Amalric M, Pin JP, Acher FC. Sibille P, et al. Among authors: oueslati n. J Med Chem. 2007 Jul 26;50(15):3585-95. doi: 10.1021/jm070262c. Epub 2007 Jun 28. J Med Chem. 2007. PMID: 17602546

3

L-(+)-2-Amino-4-thiophosphonobutyric acid (L-thioAP4), a new potent agonist of group III metabotropic glutamate receptors: increased distal acidity affords enhanced potency.

Selvam C, Goudet C, Oueslati N, Pin JP, Acher FC. Selvam C, et al. Among authors: oueslati n. J Med Chem. 2007 Sep 20;50(19):4656-64. doi: 10.1021/jm070400y. Epub 2007 Aug 28. J Med Chem. 2007. PMID: 17722902

4

A virtual screening hit reveals new possibilities for developing group III metabotropic glutamate receptor agonists.

Selvam C, Oueslati N, Lemasson IA, Brabet I, Rigault D, Courtiol T, Cesarini S, Triballeau N, Bertrand HO, Goudet C, Pin JP, Acher FC. Selvam C, et al. Among authors: oueslati n. J Med Chem. 2010 Apr 8;53(7):2797-813. doi: 10.1021/jm901523t. J Med Chem. 2010. PMID: 20218620

5

A novel selective metabotropic glutamate receptor 4 agonist reveals new possibilities for developing subtype selective ligands with therapeutic potential.

Goudet C, Vilar B, Courtiol T, Deltheil T, Bessiron T, Brabet I, Oueslati N, Rigault D, Bertrand HO, McLean H, Daniel H, Amalric M, Acher F, Pin JP. Goudet C, et al. Among authors: oueslati n. FASEB J. 2012 Apr;26(4):1682-93. doi: 10.1096/fj.11-195941. Epub 2012 Jan 5. FASEB J. 2012. PMID: 22223752

6

Activation of a dimeric metabotropic glutamate receptor by intersubunit rearrangement.

Brock C, Oueslati N, Soler S, Boudier L, Rondard P, Pin JP. Brock C, et al. Among authors: oueslati n. J Biol Chem. 2007 Nov 9;282(45):33000-8. doi: 10.1074/jbc.M702542200. Epub 2007 Sep 13. J Biol Chem. 2007. PMID: 17855348 Free article.

7

Metabotropic glutamate receptor subtype 4 selectively modulates both glutamate and GABA transmission in the striatum: implications for Parkinson's disease treatment.

Cuomo D, Martella G, Barabino E, Platania P, Vita D, Madeo G, Selvam C, Goudet C, Oueslati N, Pin JP, Acher F, Pisani A, Beurrier C, Melon C, Kerkerian-Le Goff L, Gubellini P. Cuomo D, et al. Among authors: oueslati n. J Neurochem. 2009 May;109(4):1096-105. doi: 10.1111/j.1471-4159.2009.06036.x. Epub 2009 Mar 14. J Neurochem. 2009. PMID: 19519781 Free article.

8

Time-resolved FRET strategy to screen GPCR ligand library.

Oueslati N, Hounsou C, Belhocine A, Rodriguez T, Dupuis E, Zwier JM, Trinquet E, Pin JP, Durroux T. Oueslati N, et al. Methods Mol Biol. 2015;1272:23-36. doi: 10.1007/978-1-4939-2336-6_2. Methods Mol Biol. 2015. PMID: 25563174

9

Functioning of the dimeric GABA(B) receptor extracellular domain revealed by glycan wedge scanning.

Rondard P, Huang S, Monnier C, Tu H, Blanchard B, Oueslati N, Malhaire F, Li Y, Trinquet E, Labesse G, Pin JP, Liu J. Rondard P, et al. Among authors: oueslati n. EMBO J. 2008 May 7;27(9):1321-32. doi: 10.1038/emboj.2008.64. Epub 2008 Apr 3. EMBO J. 2008. PMID: 18388862 Free PMC article.

10

Time-resolved FRET binding assay to investigate hetero-oligomer binding properties: proof of concept with dopamine D1/D3 heterodimer.

Hounsou C, Margathe JF, Oueslati N, Belhocine A, Dupuis E, Thomas C, Mann A, Ilien B, Rognan D, Trinquet E, Hibert M, Pin JP, Bonnet D, Durroux T. Hounsou C, et al. Among authors: oueslati n. ACS Chem Biol. 2015 Feb 20;10(2):466-74. doi: 10.1021/cb5007568. Epub 2014 Nov 11. ACS Chem Biol. 2015. PMID: 25350273

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