Pastorin G - Search Results

1

5,7-Disubstituted-[1,2,4]triazolo[1,5-a][1,3,5]triazines as pharmacological tools to explore the antagonist selectivity profiles toward adenosine receptors.

Federico S, Ciancetta A, Porta N, Redenti S, Pastorin G, Cacciari B, Klotz KN, Moro S, Spalluto G. Federico S, et al. Among authors: pastorin g. Eur J Med Chem. 2016 Jan 27;108:529-541. doi: 10.1016/j.ejmech.2015.12.019. Epub 2015 Dec 15. Eur J Med Chem. 2016. PMID: 26717203 Free article.

2

A facile and novel synthesis of N(2)-, C(6)-substituted pyrazolo[3,4-d]pyrimidine-4 carboxylate derivatives as adenosine receptor antagonists.

Venkatesan G, Paira P, Cheong SL, Federico S, Klotz KN, Spalluto G, Pastorin G. Venkatesan G, et al. Among authors: pastorin g. Eur J Med Chem. 2015 Mar 6;92:784-98. doi: 10.1016/j.ejmech.2015.01.046. Epub 2015 Jan 22. Eur J Med Chem. 2015. PMID: 25633494

3

Synthesis, biological activity, and molecular modeling investigation of new pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as human A(3) adenosine receptor antagonists.

Baraldi PG, Cacciari B, Moro S, Spalluto G, Pastorin G, Da Ros T, Klotz KN, Varani K, Gessi S, Borea PA. Baraldi PG, et al. Among authors: pastorin g. J Med Chem. 2002 Feb 14;45(4):770-80. doi: 10.1021/jm0109614. J Med Chem. 2002. PMID: 11831890

4

Synthesis, biological properties, and molecular modeling investigation of the first potent, selective, and water-soluble human A(3) adenosine receptor antagonist.

Maconi A, Pastorin G, Da Ros T, Spalluto G, Gao ZG, Jacobson KA, Baraldi PG, Cacciari B, Varani K, Moro S, Borea PA. Maconi A, et al. Among authors: pastorin g. J Med Chem. 2002 Aug 15;45(17):3579-82. doi: 10.1021/jm020974x. J Med Chem. 2002. PMID: 12166930 Free PMC article.

5

Pyrazolo-triazolo-pyrimidine derivatives as adenosine receptor antagonists: a possible template for adenosine receptor subtypes?

Baraldi PG, Cacciari B, Borean PA, Varanin K, Pastorin G, Da Ros T, Tabrizi MA, Fruttarolo F, Spalluto G. Baraldi PG, et al. Among authors: pastorin g. Curr Pharm Des. 2002;8(26):2299-332. doi: 10.2174/1381612023392838. Curr Pharm Des. 2002. PMID: 12369947 Review.

6

Medicinal chemistry of A2A adenosine receptor antagonists.

Cacciari B, Pastorin G, Spalluto G. Cacciari B, et al. Among authors: pastorin g. Curr Top Med Chem. 2003;3(4):403-11. doi: 10.2174/1568026033392183. Curr Top Med Chem. 2003. PMID: 12570758 Review.

7

Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor antagonists. Influence of the N5 substituent on the affinity at the human A 3 and A 2B adenosine receptor subtypes: a molecular modeling investigation.

Pastorin G, Da Ros T, Spalluto G, Deflorian F, Moro S, Cacciari B, Baraldi PG, Gessi S, Varani K, Borea PA. Pastorin G, et al. J Med Chem. 2003 Sep 25;46(20):4287-96. doi: 10.1021/jm030852k. J Med Chem. 2003. PMID: 13678407

8

Combined target-based and ligand-based drug design approach as a tool to define a novel 3D-pharmacophore model of human A3 adenosine receptor antagonists: pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as a key study.

Moro S, Braiuca P, Deflorian F, Ferrari C, Pastorin G, Cacciari B, Baraldi PG, Varani K, Borea PA, Spalluto G. Moro S, et al. Among authors: pastorin g. J Med Chem. 2005 Jan 13;48(1):152-62. doi: 10.1021/jm049662f. J Med Chem. 2005. PMID: 15634009

9

Synthesis, biological studies and molecular modeling investigation of 1,3-dimethyl-2,4-dioxo-6-methyl-8-(substituted) 1,2,3,4-tetrahydro [1,2,4]-triazolo [3,4-f]-purines as potential adenosine receptor antagonists.

Pastorin G, Bolcato C, Cacciari B, Kachler S, Klotz KN, Montopoli C, Moro S, Spalluto G. Pastorin G, et al. Farmaco. 2005 Apr;60(4):299-306. doi: 10.1016/j.farmac.2005.01.008. Farmaco. 2005. PMID: 15848204

10

A2B adenosine receptor antagonists: recent developments.

Cacciari B, Pastorin G, Bolcato C, Spalluto G, Bacilieri M, Moro S. Cacciari B, et al. Among authors: pastorin g. Mini Rev Med Chem. 2005 Dec;5(12):1053-60. doi: 10.2174/138955705774933374. Mini Rev Med Chem. 2005. PMID: 16375751 Review.

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