Podjarny A - Search Results

1

Iminosugar-Cyclopeptoid Conjugates Raise Multivalent Effect in Glycosidase Inhibition at Unprecedented High Levels.

Lepage ML, Schneider JP, Bodlenner A, Meli A, De Riccardis F, Schmitt M, Tarnus C, Nguyen-Huynh NT, Francois YN, Leize-Wagner E, Birck C, Cousido-Siah A, Podjarny A, Izzo I, Compain P. Lepage ML, et al. Among authors: podjarny a. Chemistry. 2016 Apr 4;22(15):5151-5. doi: 10.1002/chem.201600338. Epub 2016 Feb 24. Chemistry. 2016. PMID: 26917097

2

Structural Basis of Outstanding Multivalent Effects in Jack Bean α-Mannosidase Inhibition.

Howard E, Cousido-Siah A, Lepage ML, Schneider JP, Bodlenner A, Mitschler A, Meli A, Izzo I, Alvarez HA, Podjarny A, Compain P. Howard E, et al. Among authors: podjarny a. Angew Chem Int Ed Engl. 2018 Jul 2;57(27):8002-8006. doi: 10.1002/anie.201801202. Epub 2018 Jun 6. Angew Chem Int Ed Engl. 2018. PMID: 29722924

3

X-ray structure of the V301L aldo-keto reductase 1B10 complexed with NADP(+) and the potent aldose reductase inhibitor fidarestat: implications for inhibitor binding and selectivity.

Ruiz FX, Cousido-Siah A, Mitschler A, Farrés J, Parés X, Podjarny A. Ruiz FX, et al. Among authors: podjarny a. Chem Biol Interact. 2013 Feb 25;202(1-3):178-85. doi: 10.1016/j.cbi.2012.12.013. Epub 2013 Jan 4. Chem Biol Interact. 2013. PMID: 23295227

4

Crystal packing modifies ligand binding affinity: the case of aldose reductase.

Cousido-Siah A, Petrova T, Hazemann I, Mitschler A, Ruiz FX, Howard E, Ginell S, Atmanene C, Van Dorsselaer A, Sanglier-Cianférani S, Joachimiak A, Podjarny A. Cousido-Siah A, et al. Among authors: podjarny a. Proteins. 2012 Nov;80(11):2552-61. doi: 10.1002/prot.24136. Epub 2012 Jul 28. Proteins. 2012. PMID: 22752989 Free PMC article.

5

X-Ray Crystal Structure of the Full Length Human Chitotriosidase (CHIT1) Reveals Features of Its Chitin Binding Domain.

Fadel F, Zhao Y, Cousido-Siah A, Ruiz FX, Mitschler A, Podjarny A. Fadel F, et al. Among authors: podjarny a. PLoS One. 2016 Apr 25;11(4):e0154190. doi: 10.1371/journal.pone.0154190. eCollection 2016. PLoS One. 2016. PMID: 27111557 Free PMC article.

6

Probing the roles of two tryptophans surrounding the unique zinc coordination site in lipase family I.5.

Timucin E, Cousido-Siah A, Mitschler A, Podjarny A, Sezerman OU. Timucin E, et al. Among authors: podjarny a. Proteins. 2016 Jan;84(1):129-42. doi: 10.1002/prot.24961. Epub 2015 Dec 9. Proteins. 2016. PMID: 26573720

7

Validation of surface plasmon resonance screening of a diverse chemical library for the discovery of protein tyrosine phosphatase 1b binders.

Zeder-Lutz G, Choulier L, Besse M, Cousido-Siah A, Ruiz Figueras FX, Didier B, Jung ML, Podjarny A, Altschuh D. Zeder-Lutz G, et al. Among authors: podjarny a. Anal Biochem. 2012 Feb 15;421(2):417-27. doi: 10.1016/j.ab.2011.09.015. Epub 2011 Sep 29. Anal Biochem. 2012. PMID: 22037289

8

The Effect of Halogen-to-Hydrogen Bond Substitution on Human Aldose Reductase Inhibition.

Fanfrlík J, Ruiz FX, Kadlčíková A, Řezáč J, Cousido-Siah A, Mitschler A, Haldar S, Lepšík M, Kolář MH, Majer P, Podjarny AD, Hobza P. Fanfrlík J, et al. Among authors: podjarny ad. ACS Chem Biol. 2015 Jul 17;10(7):1637-42. doi: 10.1021/acschembio.5b00151. Epub 2015 May 6. ACS Chem Biol. 2015. PMID: 25919404

9

Structural analysis of sulindac as an inhibitor of aldose reductase and AKR1B10.

Cousido-Siah A, Ruiz FX, Crespo I, Porté S, Mitschler A, Parés X, Podjarny A, Farrés J. Cousido-Siah A, et al. Among authors: podjarny a. Chem Biol Interact. 2015 Jun 5;234:290-6. doi: 10.1016/j.cbi.2014.12.018. Epub 2014 Dec 20. Chem Biol Interact. 2015. PMID: 25532697

10

Design, synthesis, structure-activity relationships and X-ray structural studies of novel 1-oxopyrimido[4,5-c]quinoline-2-acetic acid derivatives as selective and potent inhibitors of human aldose reductase.

Crespo I, Giménez-Dejoz J, Porté S, Cousido-Siah A, Mitschler A, Podjarny A, Pratsinis H, Kletsas D, Parés X, Ruiz FX, Metwally K, Farrés J. Crespo I, et al. Among authors: podjarny a. Eur J Med Chem. 2018 May 25;152:160-174. doi: 10.1016/j.ejmech.2018.04.015. Epub 2018 Apr 12. Eur J Med Chem. 2018. PMID: 29705708

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