Poli S - Search Results

1

Comparison of in vitro P-glycoprotein screening assays: recommendations for their use in drug discovery.

Schwab D, Fischer H, Tabatabaei A, Poli S, Huwyler J. Schwab D, et al. Among authors: poli s. J Med Chem. 2003 Apr 24;46(9):1716-25. doi: 10.1021/jm021012t. J Med Chem. 2003. PMID: 12699389

2

An aminomethylpyrimidine DPP-IV inhibitor with improved properties.

Peters JU, Hunziker D, Fischer H, Kansy M, Weber S, Kritter S, Müller A, Wallier A, Ricklin F, Boehringer M, Poli SM, Csato M, Loeffler BM. Peters JU, et al. Among authors: poli sm. Bioorg Med Chem Lett. 2004 Jul 5;14(13):3575-8. doi: 10.1016/j.bmcl.2004.04.048. Bioorg Med Chem Lett. 2004. PMID: 15177477

3

Discovery of potent, balanced and orally active dual NK1/NK3 receptor ligands.

Peters JU, Hoffmann T, Schnider P, Stadler H, Koblet A, Alker A, Poli SM, Ballard TM, Spooren W, Steward L, Sleight AJ. Peters JU, et al. Bioorg Med Chem Lett. 2010 Jun 1;20(11):3405-8. doi: 10.1016/j.bmcl.2010.04.008. Epub 2010 Apr 9. Bioorg Med Chem Lett. 2010. PMID: 20430616

4

Influence of the 5-HT6 receptor on acetylcholine release in the cortex: pharmacological characterization of 4-(2-bromo-6-pyrrolidin-1-ylpyridine-4-sulfonyl)phenylamine, a potent and selective 5-HT6 receptor antagonist.

Riemer C, Borroni E, Levet-Trafit B, Martin JR, Poli S, Porter RH, Bös M. Riemer C, et al. Among authors: poli s. J Med Chem. 2003 Mar 27;46(7):1273-6. doi: 10.1021/jm021085c. J Med Chem. 2003. PMID: 12646038

5

Novel hexahydrospiro[piperidine-4,1'-pyrrolo[3,4-c]pyrroles]: highly selective small-molecule nociceptin/orphanin FQ receptor agonists.

Kolczewski S, Adam G, Cesura AM, Jenck F, Hennig M, Oberhauser T, Poli SM, Rössler F, Röver S, Wichmann J, Dautzenberg FM. Kolczewski S, et al. Among authors: poli sm. J Med Chem. 2003 Jan 16;46(2):255-64. doi: 10.1021/jm0209174. J Med Chem. 2003. PMID: 12519064

6

Design and synthesis of a novel, achiral class of highly potent and selective, orally active neurokinin-1 receptor antagonists.

Hoffmann T, Bös M, Stadler H, Schnider P, Hunkeler W, Godel T, Galley G, Ballard TM, Higgins GA, Poli SM, Sleight AJ. Hoffmann T, et al. Bioorg Med Chem Lett. 2006 Mar 1;16(5):1362-5. doi: 10.1016/j.bmcl.2005.11.047. Epub 2005 Dec 5. Bioorg Med Chem Lett. 2006. PMID: 16332435

7

Endogenous proteins controlling amyloid beta-peptide polymerization. Possible implications for beta-amyloid formation in the central nervous system and in peripheral tissues.

Bohrmann B, Tjernberg L, Kuner P, Poli S, Levet-Trafit B, Näslund J, Richards G, Huber W, Döbeli H, Nordstedt C. Bohrmann B, et al. Among authors: poli s. J Biol Chem. 1999 Jun 4;274(23):15990-5. doi: 10.1074/jbc.274.23.15990. J Biol Chem. 1999. PMID: 10347147 Free article.

8

Cytochrome p450 enzymes mechanism based inhibitors: common sub-structures and reactivity.

Fontana E, Dansette PM, Poli SM. Fontana E, et al. Among authors: poli sm. Curr Drug Metab. 2005 Oct;6(5):413-54. doi: 10.2174/138920005774330639. Curr Drug Metab. 2005. PMID: 16248836 Review.

9

A novel series of metabotropic glutamate receptor 5 negative allosteric modulators based on a 4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine core.

Duvey G, Perry B, Le Poul E, Poli S, Bonnet B, Lambeng N, Charvin D, Donovan-Rodrigues T, Haddouk H, Gagliardi S, Rocher JP. Duvey G, et al. Among authors: poli s. Bioorg Med Chem Lett. 2013 Aug 15;23(16):4523-7. doi: 10.1016/j.bmcl.2013.06.044. Epub 2013 Jun 25. Bioorg Med Chem Lett. 2013. PMID: 23850200

10

Discovery of 1,4-disubstituted 3-cyano-2-pyridones: a new class of positive allosteric modulators of the metabotropic glutamate 2 receptor.

Cid JM, Duvey G, Tresadern G, Nhem V, Furnari R, Cluzeau P, Vega JA, de Lucas AI, Matesanz E, Alonso JM, Linares ML, Andrés JI, Poli SM, Lutjens R, Himogai H, Rocher JP, Macdonald GJ, Oehlrich D, Lavreysen H, Ahnaou A, Drinkenburg W, Mackie C, Trabanco AA. Cid JM, et al. J Med Chem. 2012 Mar 8;55(5):2388-405. doi: 10.1021/jm2016864. Epub 2012 Feb 24. J Med Chem. 2012. PMID: 22364337

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