Rochel N - Search Results

1

Superagonistic action of 14-epi-analogs of 1,25-dihydroxyvitamin D explained by vitamin D receptor-coactivator interaction.

Eelen G, Verlinden L, Rochel N, Claessens F, De Clercq P, Vandewalle M, Tocchini-Valentini G, Moras D, Bouillon R, Verstuyf A. Eelen G, et al. Among authors: rochel n. Mol Pharmacol. 2005 May;67(5):1566-73. doi: 10.1124/mol.104.008730. Epub 2005 Feb 22. Mol Pharmacol. 2005. PMID: 15728261

2

Further Studies on the Highly Active Des-C-Ring and Aromatic-D-Ring Analogues of 1α,25-Dihydroxyvitamin D₃ (Calcitriol): Refinement of the Side Chain.

Zárate-Ruíz A, Seoane S, Peluso-Iltis C, Peters S, Gregorio C, Guiberteau T, Maestro M, Pérez-Fernández R, Rochel N, Mouriño A. Zárate-Ruíz A, et al. Among authors: rochel n. J Med Chem. 2023 Nov 23;66(22):15326-15339. doi: 10.1021/acs.jmedchem.3c01371. Epub 2023 Nov 1. J Med Chem. 2023. PMID: 37910811

3

Vitamin D Receptor Antagonist MeTC7 Inhibits PD-L1.

Khazan N, Quarato ER, Singh NA, Snyder CWA, Moore T, Miller JP, Yasui M, Teramoto Y, Goto T, Reshi S, Hong J, Zhang N, Pandey D, Srivastava P, Morell A, Kawano H, Kawano Y, Conley T, Sahasrabudhe DM, Yano N, Miyamoto H, Aljitawi O, Liesveld J, Becker MW, Calvi LM, Zhovmer AS, Tabdanov ED, Dokholyan NV, Linehan DC, Hansen JN, Gerber SA, Sharon A, Khera MK, Jurutka PW, Rochel N, Kim KK, Rowswell-Turner RB, Singh RK, Moore RG. Khazan N, et al. Among authors: rochel n. Cancers (Basel). 2023 Jun 30;15(13):3432. doi: 10.3390/cancers15133432. Cancers (Basel). 2023. PMID: 37444542 Free PMC article.

4

Large-scale expression and purification of the human vitamin D receptor and its ligand-binding domain for structural studies.

Juntunen K, Rochel N, Moras D, Vihko P. Juntunen K, et al. Among authors: rochel n. Biochem J. 1999 Dec 1;344 Pt 2(Pt 2):297-303. Biochem J. 1999. PMID: 10567209 Free PMC article.

5

The crystal structure of the nuclear receptor for vitamin D bound to its natural ligand.

Rochel N, Wurtz JM, Mitschler A, Klaholz B, Moras D. Rochel N, et al. Mol Cell. 2000 Jan;5(1):173-9. doi: 10.1016/s1097-2765(00)80413-x. Mol Cell. 2000. PMID: 10678179 Free article.

6

Functional and structural characterization of the insertion region in the ligand binding domain of the vitamin D nuclear receptor.

Rochel N, Tocchini-Valentini G, Egea PF, Juntunen K, Garnier JM, Vihko P, Moras D. Rochel N, et al. Eur J Biochem. 2001 Feb;268(4):971-9. doi: 10.1046/j.1432-1327.2001.01953.x. Eur J Biochem. 2001. PMID: 11179963 Free article.

7

Effects of ligand binding on the association properties and conformation in solution of retinoic acid receptors RXR and RAR.

Egea PF, Rochel N, Birck C, Vachette P, Timmins PA, Moras D. Egea PF, et al. Among authors: rochel n. J Mol Biol. 2001 Mar 23;307(2):557-76. doi: 10.1006/jmbi.2000.4409. J Mol Biol. 2001. PMID: 11254382

8

Crystal structures of the vitamin D receptor complexed to superagonist 20-epi ligands.

Tocchini-Valentini G, Rochel N, Wurtz JM, Mitschler A, Moras D. Tocchini-Valentini G, et al. Among authors: rochel n. Proc Natl Acad Sci U S A. 2001 May 8;98(10):5491-6. doi: 10.1073/pnas.091018698. Proc Natl Acad Sci U S A. 2001. PMID: 11344298 Free PMC article.

9

Structural adaptability in the ligand-binding pocket of the ecdysone hormone receptor.

Billas IM, Iwema T, Garnier JM, Mitschler A, Rochel N, Moras D. Billas IM, et al. Among authors: rochel n. Nature. 2003 Nov 6;426(6962):91-6. doi: 10.1038/nature02112. Epub 2003 Nov 2. Nature. 2003. PMID: 14595375

10

Crystal structures of the vitamin D nuclear receptor liganded with the vitamin D side chain analogues calcipotriol and seocalcitol, receptor agonists of clinical importance. Insights into a structural basis for the switching of calcipotriol to a receptor antagonist by further side chain modification.

Tocchini-Valentini G, Rochel N, Wurtz JM, Moras D. Tocchini-Valentini G, et al. Among authors: rochel n. J Med Chem. 2004 Apr 8;47(8):1956-61. doi: 10.1021/jm0310582. J Med Chem. 2004. PMID: 15055995

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