S10 OD021734/OD/NIH HHS/United States[Grant Number] - Search Results

Year	Number of Results
2015	1
2016	2
2017	2
2018	6
2019	11
2020	4
2021	3
2022	6
2023	6
2024	0

1

Design, synthesis, and biological evaluation of a novel series of 1,2,4-oxadiazole inhibitors of SLACK potassium channels: Identification of in vitro tool VU0935685.

Qunies AM, Spitznagel BD, Du Y, David Weaver C, Emmitte KA. Qunies AM, et al. Bioorg Med Chem. 2023 Nov 15;95:117487. doi: 10.1016/j.bmc.2023.117487. Epub 2023 Sep 30. Bioorg Med Chem. 2023. PMID: 37812884

2

Arrest of mouse preterm labor until term delivery by combination therapy with atosiban and mundulone, a natural product with tocolytic efficacy.

Siricilla S, Hansen CJ, Rogers JH, De D, Simpson CL, Waterson AG, Sulikowski GA, Crockett SL, Boatwright N, Reese J, Paria BC, Newton J, Herington JL. Siricilla S, et al. Pharmacol Res. 2023 Sep;195:106876. doi: 10.1016/j.phrs.2023.106876. Epub 2023 Aug 1. Pharmacol Res. 2023. PMID: 37536638 Free PMC article.

3

Small Molecule Activation of NAPE-PLD Enhances Efferocytosis by Macrophages.

Zarrow JE, Alli-Oluwafuyi AM, Youwakim CM, Kim K, Jenkins AN, Suero IC, Jones MR, Mashhadi Z, Mackie K, Waterson AG, Doran AC, Sulikowski GA, Davies SS. Zarrow JE, et al. ACS Chem Biol. 2023 Aug 18;18(8):1891-1904. doi: 10.1021/acschembio.3c00401. Epub 2023 Aug 2. ACS Chem Biol. 2023. PMID: 37531659 Free article.

4

Synthesis and SAR of a novel Kir6.2/SUR1 channel opener scaffold identified by HTS.

Dodd CJ, Chronister KS, Rathnayake U, Parr LC, Li K, Chang S, Mi D, Days EL, Bauer JA, Cho HP, Boutaud O, Denton JS, Lindsley CW, Han C. Dodd CJ, et al. Bioorg Med Chem Lett. 2023 May 1;87:129256. doi: 10.1016/j.bmcl.2023.129256. Epub 2023 Mar 24. Bioorg Med Chem Lett. 2023. PMID: 36966977

5

Identification of Potent, Selective, and Peripherally Restricted Serotonin Receptor 2B Antagonists from a High-Throughput Screen.

Bender AM, Valentine MS, Bauer JA, Days E, Lindsley CW, Merryman WD. Bender AM, et al. Assay Drug Dev Technol. 2023 Apr;21(3):89-96. doi: 10.1089/adt.2022.116. Epub 2023 Mar 17. Assay Drug Dev Technol. 2023. PMID: 36930852 Free PMC article.

6

Small Molecule Activation of NAPE-PLD Enhances Efferocytosis by Macrophages.

Zarrow JE, Alli-Oluwafuyi AM, Youwakim CM, Kim K, Jenkins AN, Suero IC, Jones MR, Mashhadi Z, Mackie KP, Waterson AG, Doran AC, Sulikowski GA, Davies SS. Zarrow JE, et al. bioRxiv [Preprint]. 2023 Feb 28:2023.01.25.525554. doi: 10.1101/2023.01.25.525554. bioRxiv. 2023. PMID: 36747693 Free PMC article. Updated. Preprint.

7

Structure-activity relationship studies in a new series of 2-amino-N-phenylacetamide inhibitors of Slack potassium channels.

Qunies AM, Mishra NM, Spitznagel BD, Du Y, Acuña VS, David Weaver C, Emmitte KA. Qunies AM, et al. Bioorg Med Chem Lett. 2022 Nov 15;76:129013. doi: 10.1016/j.bmcl.2022.129013. Epub 2022 Sep 29. Bioorg Med Chem Lett. 2022. PMID: 36184030 Free PMC article.

8

A BRET Ca²⁺ sensor enables high-throughput screening in the presence of background fluorescence.

Cumberbatch D, Mori T, Yang J, Mi D, Vinson P, Weaver CD, Johnson CH. Cumberbatch D, et al. Sci Signal. 2022 Aug 16;15(747):eabq7618. doi: 10.1126/scisignal.abq7618. Epub 2022 Aug 16. Sci Signal. 2022. PMID: 35973028 Free PMC article.

9

Discovery of Small Molecule KCC2 Potentiators Which Attenuate In Vitro Seizure-Like Activity in Cultured Neurons.

Prael Iii FJ, Kim K, Du Y, Spitznagel BD, Sulikowski GA, Delpire E, Weaver CD. Prael Iii FJ, et al. Front Cell Dev Biol. 2022 Jun 24;10:912812. doi: 10.3389/fcell.2022.912812. eCollection 2022. Front Cell Dev Biol. 2022. PMID: 35813195 Free PMC article.

10

Development of VU6019650: A Potent, Highly Selective, and Systemically Active Orthosteric Antagonist of the M₅ Muscarinic Acetylcholine Receptor for the Treatment of Opioid Use Disorder.

Garrison AT, Orsi DL, Capstick RA, Whomble D, Li J, Carter TR, Felts AS, Vinson PN, Rodriguez AL, Han A, Hajari K, Cho HP, Teal LB, Ragland MG, Ghamari-Langroudi M, Bubser M, Chang S, Schnetz-Boutaud NC, Boutaud O, Blobaum AL, Foster DJ, Niswender CM, Conn PJ, Lindsley CW, Jones CK, Han C. Garrison AT, et al. J Med Chem. 2022 Apr 28;65(8):6273-6286. doi: 10.1021/acs.jmedchem.2c00192. Epub 2022 Apr 13. J Med Chem. 2022. PMID: 35417155

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