Sakamuri S - Search Results

1

Discovery of a novel dopamine transporter inhibitor, 4-hydroxy-1-methyl-4-(4-methylphenyl)-3-piperidyl 4-methylphenyl ketone, as a potential cocaine antagonist through 3D-database pharmacophore searching. Molecular modeling, structure-activity relationships, and behavioral pharmacological studies.

Wang S, Sakamuri S, Enyedy IJ, Kozikowski AP, Deschaux O, Bandyopadhyay BC, Tella SR, Zaman WA, Johnson KM. Wang S, et al. Among authors: sakamuri s. J Med Chem. 2000 Feb 10;43(3):351-60. doi: 10.1021/jm990516x. J Med Chem. 2000. PMID: 10669562

2

2,3-Disubstituted quinuclidines as a novel class of dopamine transporter inhibitors.

Sakamuri S, Enyedy IJ, Zaman WA, Tella SR, Kozikowski AP, Flippen-Anderson JL, Farkas T, Johnson KM, Wang S. Sakamuri S, et al. Bioorg Med Chem. 2003 Mar 20;11(6):1123-36. doi: 10.1016/s0968-0896(02)00450-9. Bioorg Med Chem. 2003. PMID: 12614900

3

Pharmacophore-based discovery of substituted pyridines as novel dopamine transporter inhibitors.

Enyedy IJ, Sakamuri S, Zaman WA, Johnson KM, Wang S. Enyedy IJ, et al. Among authors: sakamuri s. Bioorg Med Chem Lett. 2003 Feb 10;13(3):513-7. doi: 10.1016/s0960-894x(02)00943-5. Bioorg Med Chem Lett. 2003. PMID: 12565962

4

Pharmacophore-based discovery, synthesis, and biological evaluation of 4-phenyl-1-arylalkyl piperidines as dopamine transporter inhibitors.

Sakamuri S, Enyedy IJ, Kozikowski AP, Zaman WA, Johnson KM, Wang S. Sakamuri S, et al. Bioorg Med Chem Lett. 2001 Feb 26;11(4):495-500. doi: 10.1016/s0960-894x(00)00703-4. Bioorg Med Chem Lett. 2001. PMID: 11229756

5

Pharmacophore-based discovery of 3,4-disubstituted pyrrolidines as a novel class of monoamine transporter inhibitors.

Enyedy IJ, Zaman WA, Sakamuri S, Kozikowski AP, Johnson KM, Wang S. Enyedy IJ, et al. Among authors: sakamuri s. Bioorg Med Chem Lett. 2001 May 7;11(9):1113-8. doi: 10.1016/s0960-894x(01)00132-9. Bioorg Med Chem Lett. 2001. PMID: 11354356

6

Molecular modeling, structure--activity relationships and functional antagonism studies of 4-hydroxy-1-methyl-4-(4-methylphenyl)-3-piperidyl 4-methylphenyl ketones as a novel class of dopamine transporter inhibitors.

Wang S, Sakamuri S, Enyedy IJ, Kozikowski AP, Zaman WA, Johnson KM. Wang S, et al. Among authors: sakamuri s. Bioorg Med Chem. 2001 Jul;9(7):1753-64. doi: 10.1016/s0968-0896(01)00090-6. Bioorg Med Chem. 2001. PMID: 11425577

7

Synthesis and modeling study of (2S,5R,6R)- and (2S,5R,6S)-6-hydroxy- 8-(1-decynyl)-benzolactam-V8 as protein kinase C modulators.

Wei ZL, Sakamuri S, Petukhov PA, George C, Lewin NE, Blumberg PM, Kozikowski AP. Wei ZL, et al. Among authors: sakamuri s. Org Lett. 2002 Jun 27;4(13):2169-72. doi: 10.1021/ol026013u. Org Lett. 2002. PMID: 12074659

8

Solution phase parallel synthesis and evaluation of MAPK inhibitory activities of close structural analogues of a Ras pathway modulator.

Lu Y, Sakamuri S, Chen QZ, Keng YF, Khazak V, Illgen K, Schabbert S, Weber L, Menon SR. Lu Y, et al. Among authors: sakamuri s. Bioorg Med Chem Lett. 2004 Aug 2;14(15):3957-62. doi: 10.1016/j.bmcl.2004.05.048. Bioorg Med Chem Lett. 2004. PMID: 15225706

9

Design and modular parallel synthesis of a MCR derived alpha-helix mimetic protein-protein interaction inhibitor scaffold.

Antuch W, Menon S, Chen QZ, Lu Y, Sakamuri S, Beck B, Schauer-Vukasinović V, Agarwal S, Hess S, Dömling A. Antuch W, et al. Among authors: sakamuri s. Bioorg Med Chem Lett. 2006 Mar 15;16(6):1740-3. doi: 10.1016/j.bmcl.2005.11.102. Epub 2006 Jan 19. Bioorg Med Chem Lett. 2006. PMID: 16427279

10

Inhibitors of Ras/Raf-1 interaction identified by two-hybrid screening revert Ras-dependent transformation phenotypes in human cancer cells.

Kato-Stankiewicz J, Hakimi I, Zhi G, Zhang J, Serebriiskii I, Guo L, Edamatsu H, Koide H, Menon S, Eckl R, Sakamuri S, Lu Y, Chen QZ, Agarwal S, Baumbach WR, Golemis EA, Tamanoi F, Khazak V. Kato-Stankiewicz J, et al. Among authors: sakamuri s. Proc Natl Acad Sci U S A. 2002 Oct 29;99(22):14398-403. doi: 10.1073/pnas.222222699. Epub 2002 Oct 21. Proc Natl Acad Sci U S A. 2002. PMID: 12391290 Free PMC article.

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