Scozzafava A - Search Results

1

Tricyclic sulfonamides incorporating benzothiopyrano[4,3-c]pyrazole and pyridothiopyrano[4,3-c]pyrazole effectively inhibit α- and β-carbonic anhydrase: X-ray crystallography and solution investigations on 15 isoforms.

Marini AM, Maresca A, Aggarwal M, Orlandini E, Nencetti S, Da Settimo F, Salerno S, Simorini F, La Motta C, Taliani S, Nuti E, Scozzafava A, McKenna R, Rossello A, Supuran CT. Marini AM, et al. Among authors: scozzafava a. J Med Chem. 2012 Nov 26;55(22):9619-29. doi: 10.1021/jm300878g. Epub 2012 Nov 8. J Med Chem. 2012. PMID: 23067387

2

Carbonic anhydrase activators: high affinity isozymes I, II, and IV activators, incorporating a beta-alanyl-histidine scaffold.

Scozzafava A, Supuran CT. Scozzafava A, et al. J Med Chem. 2002 Jan 17;45(2):284-91. doi: 10.1021/jm010958k. J Med Chem. 2002. PMID: 11784133

3

Carbonic anhydrase inhibitors. A general approach for the preparation of water-soluble sulfonamides incorporating polyamino-polycarboxylate tails and of their metal complexes possessing long-lasting, topical intraocular pressure-lowering properties.

Scozzafava A, Menabuoni L, Mincione F, Supuran CT. Scozzafava A, et al. J Med Chem. 2002 Mar 28;45(7):1466-76. doi: 10.1021/jm0108202. J Med Chem. 2002. PMID: 11906288

4

Carbonic anhydrase activators: human isozyme II is strongly activated by oligopeptides incorporating the carboxyterminal sequence of the bicarbonate anion exchanger AE1.

Scozzafava A, Supuran CT. Scozzafava A, et al. Bioorg Med Chem Lett. 2002 Apr 22;12(8):1177-80. doi: 10.1016/s0960-894x(02)00121-x. Bioorg Med Chem Lett. 2002. PMID: 11934582

5

Carbonic anhydrase inhibitors. Preparation of potent sulfonamides inhibitors incorporating bile acid tails.

Scozzafava A, Supuran CT. Scozzafava A, et al. Bioorg Med Chem Lett. 2002 Jun 17;12(12):1551-7. doi: 10.1016/s0960-894x(02)00252-4. Bioorg Med Chem Lett. 2002. PMID: 12039560

6

Nonaromatic sulfonamide group as an ideal anchor for potent human carbonic anhydrase inhibitors: role of hydrogen-bonding networks in ligand binding and drug design.

Abbate F, Supuran CT, Scozzafava A, Orioli P, Stubbs MT, Klebe G. Abbate F, et al. Among authors: scozzafava a. J Med Chem. 2002 Aug 15;45(17):3583-7. doi: 10.1021/jm011131t. J Med Chem. 2002. PMID: 12166931

7

Carbonic anhydrase inhibitors.

Supuran CT, Scozzafava A, Casini A. Supuran CT, et al. Among authors: scozzafava a. Med Res Rev. 2003 Mar;23(2):146-89. doi: 10.1002/med.10025. Med Res Rev. 2003. PMID: 12500287 Review.

8

Carbonic anhydrase inhibitors: inhibition of cytosolic isozymes I and II with sulfamide derivatives.

Casini A, Winum JY, Montero JL, Scozzafava A, Supuran CT. Casini A, et al. Among authors: scozzafava a. Bioorg Med Chem Lett. 2003 Mar 10;13(5):837-40. doi: 10.1016/s0960-894x(03)00028-3. Bioorg Med Chem Lett. 2003. PMID: 12617903

9

Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with aromatic and heterocyclic sulfonamides.

Vullo D, Franchi M, Gallori E, Pastorek J, Scozzafava A, Pastorekova S, Supuran CT. Vullo D, et al. Among authors: scozzafava a. Bioorg Med Chem Lett. 2003 Mar 24;13(6):1005-9. doi: 10.1016/s0960-894x(03)00091-x. Bioorg Med Chem Lett. 2003. PMID: 12643899

10

Anticancer and antiviral sulfonamides.

Scozzafava A, Owa T, Mastrolorenzo A, Supuran CT. Scozzafava A, et al. Curr Med Chem. 2003 Jun;10(11):925-53. doi: 10.2174/0929867033457647. Curr Med Chem. 2003. PMID: 12678681 Review.

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