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Acetoxymethyl Ester of Tetrabromobenzimidazole-Peptoid Conjugate for Inhibition of Protein Kinase CK2 in Living Cells.
Bioconjug Chem. 2015 Dec 16;26(12):2324-35. doi: 10.1021/acs.bioconjchem.5b00383. Epub 2015 Nov 12.
Bioconjug Chem. 2015.
PMID: 26559659
Inhibition of CREB phosphorylation by conjugates of adenosine analogues and arginine-rich peptides, inhibitors of PKA catalytic subunit.
Kriisa M, Sinijärv H, Vaasa A, Enkvist E, Kostenko S, Moens U, Uri A.
Kriisa M, et al. Among authors: sinijarv h.
Chembiochem. 2015 Jan 19;16(2):312-9. doi: 10.1002/cbic.201402526. Epub 2014 Dec 8.
Chembiochem. 2015.
PMID: 25487811
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Binding assay for characterization of protein kinase inhibitors possessing sub-picomolar to sub-millimolar affinity.
Sinijarv H, Wu S, Ivan T, Laasfeld T, Viht K, Uri A.
Sinijarv H, et al.
Anal Biochem. 2017 Aug 15;531:67-77. doi: 10.1016/j.ab.2017.05.017. Epub 2017 May 18.
Anal Biochem. 2017.
PMID: 28527909
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Competitive ligands facilitate dissociation of the complex of bifunctional inhibitor and protein kinase.
Ivan T, Enkvist E, Sinijarv H, Uri A.
Ivan T, et al. Among authors: sinijarv h.
Biophys Chem. 2017 Sep;228:17-24. doi: 10.1016/j.bpc.2017.06.004. Epub 2017 Jun 20.
Biophys Chem. 2017.
PMID: 28651101
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