Stachel SJ - Search Results

1

The fluorescence of scorpions and cataractogenesis.

Stachel SJ, Stockwell SA, Van Vranken DL. Stachel SJ, et al. Chem Biol. 1999 Aug;6(8):531-9. doi: 10.1016/S1074-5521(99)80085-4. Chem Biol. 1999. PMID: 10421760

2

Stabilization of a C7 equatorial gamma turn in DMSO-d6 by a ditryptophan crosslink.

Stachel SJ, Hu H, Van QN, Shaka AJ, Van Vranken DL. Stachel SJ, et al. Bioorg Med Chem. 1998 Sep;6(9):1439-46. doi: 10.1016/s0968-0896(98)00076-5. Bioorg Med Chem. 1998. PMID: 9801815

3

Fluorogenic peptide sequences--transformation of short peptides into fluorophores under ambient photooxidative conditions.

Juskowiak GL, Stachel SJ, Tivitmahaisoon P, Van Vranken DL. Juskowiak GL, et al. Among authors: stachel sj. J Am Chem Soc. 2004 Jan 21;126(2):550-6. doi: 10.1021/ja0379971. J Am Chem Soc. 2004. PMID: 14719952

4

Insights into long-range structural effects on the stereochemistry of aldol condensations: a practical total synthesis of desoxyepothilone F.

Lee CB, Wu Z, Zhang F, Chappell MD, Stachel SJ, Chou TC, Guan Y, Danishefsky SJ. Lee CB, et al. Among authors: stachel sj. J Am Chem Soc. 2001 Jun 6;123(22):5249-59. doi: 10.1021/ja010039j. J Am Chem Soc. 2001. PMID: 11457387

5

Concise asymmetric syntheses of radicicol and monocillin I.

Garbaccio RM, Stachel SJ, Baeschlin DK, Danishefsky SJ. Garbaccio RM, et al. Among authors: stachel sj. J Am Chem Soc. 2001 Nov 7;123(44):10903-8. doi: 10.1021/ja011364+. J Am Chem Soc. 2001. PMID: 11686693

6

Identification of a small molecule nonpeptide active site beta-secretase inhibitor that displays a nontraditional binding mode for aspartyl proteases.

Coburn CA, Stachel SJ, Li YM, Rush DM, Steele TG, Chen-Dodson E, Holloway MK, Xu M, Huang Q, Lai MT, DiMuzio J, Crouthamel MC, Shi XP, Sardana V, Chen Z, Munshi S, Kuo L, Makara GM, Annis DA, Tadikonda PK, Nash HM, Vacca JP, Wang T. Coburn CA, et al. Among authors: stachel sj. J Med Chem. 2004 Dec 2;47(25):6117-9. doi: 10.1021/jm049388p. J Med Chem. 2004. PMID: 15566281

7

Structure-based design of potent and selective cell-permeable inhibitors of human beta-secretase (BACE-1).

Stachel SJ, Coburn CA, Steele TG, Jones KG, Loutzenhiser EF, Gregro AR, Rajapakse HA, Lai MT, Crouthamel MC, Xu M, Tugusheva K, Lineberger JE, Pietrak BL, Espeseth AS, Shi XP, Chen-Dodson E, Holloway MK, Munshi S, Simon AJ, Kuo L, Vacca JP. Stachel SJ, et al. J Med Chem. 2004 Dec 16;47(26):6447-50. doi: 10.1021/jm049379g. J Med Chem. 2004. PMID: 15588077

8

Conformationally biased P3 amide replacements of beta-secretase inhibitors.

Stachel SJ, Coburn CA, Steele TG, Crouthamel MC, Pietrak BL, Lai MT, Holloway MK, Munshi SK, Graham SL, Vacca JP. Stachel SJ, et al. Bioorg Med Chem Lett. 2006 Feb;16(3):641-4. doi: 10.1016/j.bmcl.2005.10.032. Epub 2005 Nov 2. Bioorg Med Chem Lett. 2006. PMID: 16263281

9

BACE-1 inhibition by a series of psi[CH2NH] reduced amide isosteres.

Coburn CA, Stachel SJ, Jones KG, Steele TG, Rush DM, DiMuzio J, Pietrak BL, Lai MT, Huang Q, Lineberger J, Jin L, Munshi S, Katharine Holloway M, Espeseth A, Simon A, Hazuda D, Graham SL, Vacca JP. Coburn CA, et al. Among authors: stachel sj. Bioorg Med Chem Lett. 2006 Jul 15;16(14):3635-8. doi: 10.1016/j.bmcl.2006.04.076. Epub 2006 May 11. Bioorg Med Chem Lett. 2006. PMID: 16690314

10

Macrocyclic inhibitors of beta-secretase: functional activity in an animal model.

Stachel SJ, Coburn CA, Sankaranarayanan S, Price EA, Wu G, Crouthamel M, Pietrak BL, Huang Q, Lineberger J, Espeseth AS, Jin L, Ellis J, Holloway MK, Munshi S, Allison T, Hazuda D, Simon AJ, Graham SL, Vacca JP. Stachel SJ, et al. J Med Chem. 2006 Oct 19;49(21):6147-50. doi: 10.1021/jm060884i. J Med Chem. 2006. PMID: 17034118

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