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Diazinones as P2 replacements for pyrazole-based cathepsin S inhibitors.
Ameriks MK, Bembenek SD, Burdett MT, Choong IC, Edwards JP, Gebauer D, Gu Y, Karlsson L, Purkey HE, Staker BL, Sun S, Thurmond RL, Zhu J. Ameriks MK, et al. Among authors: staker bl. Bioorg Med Chem Lett. 2010 Jul 15;20(14):4060-4. doi: 10.1016/j.bmcl.2010.05.086. Epub 2010 May 25. Bioorg Med Chem Lett. 2010. PMID: 20541404
Identification of potent and selective N-myristoyltransferase inhibitors of Plasmodium vivax liver stage hypnozoites and schizonts.
Rodríguez-Hernández D, Vijayan K, Zigweid R, Fenwick MK, Sankaran B, Roobsoong W, Sattabongkot J, Glennon EKK, Myler PJ, Sunnerhagen P, Staker BL, Kaushansky A, Grøtli M. Rodríguez-Hernández D, et al. Among authors: staker bl. Nat Commun. 2023 Sep 5;14(1):5408. doi: 10.1038/s41467-023-41119-7. Nat Commun. 2023. PMID: 37669940 Free PMC article.
Active site in RrmJ, a heat shock-induced methyltransferase.
Hager J, Staker BL, Bugl H, Jakob U. Hager J, et al. Among authors: staker bl. J Biol Chem. 2002 Nov 1;277(44):41978-86. doi: 10.1074/jbc.M205423200. Epub 2002 Aug 13. J Biol Chem. 2002. PMID: 12181314 Free article.
Identification of and Structural Insights into Hit Compounds Targeting N-Myristoyltransferase for Cryptosporidium Drug Development.
Fenwick MK, Reers AR, Liu Y, Zigweid R, Sankaran B, Shin J, Hulverson MA, Hammerson B, Fernández Álvaro E, Myler PJ, Kaushansky A, Van Voorhis WC, Fan E, Staker BL. Fenwick MK, et al. Among authors: staker bl. ACS Infect Dis. 2023 Oct 13;9(10):1821-1833. doi: 10.1021/acsinfecdis.3c00151. Epub 2023 Sep 18. ACS Infect Dis. 2023. PMID: 37722671 Free PMC article.
Characterization of a family I inorganic pyrophosphatase from Legionella pneumophila Philadelphia 1.
Moorefield J, Konuk Y, Norman JO, Abendroth J, Edwards TE, Lorimer DD, Mayclin SJ, Staker BL, Craig JK, Barett KF, Barrett LK, Van Voorhis WC, Myler PJ, McLaughlin KJ. Moorefield J, et al. Among authors: staker bl. Acta Crystallogr F Struct Biol Commun. 2023 Oct 1;79(Pt 10):257-266. doi: 10.1107/S2053230X23008002. Epub 2023 Sep 20. Acta Crystallogr F Struct Biol Commun. 2023. PMID: 37728609
High-resolution crystal structure and chemical screening reveal pantothenate kinase as a new target for antifungal development.
Gihaz S, Gareiss P, Choi JY, Renard I, Pal AC, Surovsteva Y, Chiu JE, Thekkiniath J, Plummer M, Hungerford W, Montgomery ML, Hosford A, Adams EM, Lightfoot JD, Fox D 3rd, Ojo KK, Staker BL, Fuller K, Ben Mamoun C. Gihaz S, et al. Among authors: staker bl. Structure. 2022 Nov 3;30(11):1494-1507.e6. doi: 10.1016/j.str.2022.09.001. Epub 2022 Sep 26. Structure. 2022. PMID: 36167065 Free PMC article.
99 results