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Polyamines inhibit carbonic anhydrases by anchoring to the zinc-coordinated water molecule.
Carta F, Temperini C, Innocenti A, Scozzafava A, Kaila K, Supuran CT. Carta F, et al. Among authors: temperini c. J Med Chem. 2010 Aug 12;53(15):5511-22. doi: 10.1021/jm1003667. J Med Chem. 2010. PMID: 20590092
Structure-Based Identification of Inhibitory Fragments Targeting the p300/CBP-Associated Factor Bromodomain.
Chaikuad A, Lang S, Brennan PE, Temperini C, Fedorov O, Hollander J, Nachane R, Abell C, Müller S, Siegal G, Knapp S. Chaikuad A, et al. Among authors: temperini c. J Med Chem. 2016 Feb 25;59(4):1648-53. doi: 10.1021/acs.jmedchem.5b01719. Epub 2016 Jan 13. J Med Chem. 2016. PMID: 26731131 Free PMC article.
An inhibitor-like binding mode of a carbonic anhydrase activator within the active site of isoform II.
Dave K, Ilies MA, Scozzafava A, Temperini C, Vullo D, Supuran CT. Dave K, et al. Among authors: temperini c. Bioorg Med Chem Lett. 2011 May 1;21(9):2764-8. doi: 10.1016/j.bmcl.2010.10.045. Epub 2010 Oct 14. Bioorg Med Chem Lett. 2011. PMID: 21036610
Synthesis and crystallographic analysis of new sulfonamides incorporating NO-donating moieties with potent antiglaucoma action.
Mincione F, Benedini F, Biondi S, Cecchi A, Temperini C, Formicola G, Pacileo I, Scozzafava A, Masini E, Supuran CT. Mincione F, et al. Among authors: temperini c. Bioorg Med Chem Lett. 2011 Jun 1;21(11):3216-21. doi: 10.1016/j.bmcl.2011.04.046. Epub 2011 Apr 20. Bioorg Med Chem Lett. 2011. PMID: 21549597
Nitric oxide-donating carbonic anhydrase inhibitors for the treatment of open-angle glaucoma.
Steele RM, Benedini F, Biondi S, Borghi V, Carzaniga L, Impagnatiello F, Miglietta D, Chong WK, Rajapakse R, Cecchi A, Temperini C, Supuran CT. Steele RM, et al. Bioorg Med Chem Lett. 2009 Dec 1;19(23):6565-70. doi: 10.1016/j.bmcl.2009.10.036. Epub 2009 Oct 13. Bioorg Med Chem Lett. 2009. PMID: 19854054
Carbonic anhydrase activation and the drug design.
Temperini C, Scozzafava A, Supuran CT. Temperini C, et al. Curr Pharm Des. 2008;14(7):708-15. doi: 10.2174/138161208783877857. Curr Pharm Des. 2008. PMID: 18336317 Review.
Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides.
Saczewski F, Innocenti A, Sławiński J, Kornicka A, Brzozowski Z, Pomarnacka E, Scozzafava A, Temperini C, Supuran CT. Saczewski F, et al. Bioorg Med Chem. 2008 Apr 1;16(7):3933-40. doi: 10.1016/j.bmc.2008.01.034. Epub 2008 Jan 26. Bioorg Med Chem. 2008. PMID: 18242998
Carbonic anhydrase inhibitors: clash with Ala65 as a means for designing inhibitors with low affinity for the ubiquitous isozyme II, exemplified by the crystal structure of the topiramate sulfamide analogue.
Winum JY, Temperini C, El Cheikh K, Innocenti A, Vullo D, Ciattini S, Montero JL, Scozzafava A, Supuran CT. Winum JY, et al. J Med Chem. 2006 Nov 30;49(24):7024-31. doi: 10.1021/jm060807n. J Med Chem. 2006. PMID: 17125255
Carbonic anhydrase activators: L-Adrenaline plugs the active site entrance of isozyme II, activating better isoforms I, IV, VA, VII, and XIV.
Temperini C, Innocenti A, Scozzafava A, Mastrolorenzo A, Supuran CT. Temperini C, et al. Bioorg Med Chem Lett. 2007 Feb 1;17(3):628-35. doi: 10.1016/j.bmcl.2006.11.027. Epub 2006 Nov 15. Bioorg Med Chem Lett. 2007. PMID: 17127057
Carbonic anhydrase inhibitors. Interaction of 2-(hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide with 12 mammalian isoforms: kinetic and X-ray crystallographic studies.
Güzel O, Temperini C, Innocenti A, Scozzafava A, Salman A, Supuran CT. Güzel O, et al. Bioorg Med Chem Lett. 2008 Jan 1;18(1):152-8. doi: 10.1016/j.bmcl.2007.10.110. Epub 2007 Nov 4. Bioorg Med Chem Lett. 2008. PMID: 18024029
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