Triballeau N - Search Results

1

A virtual screening hit reveals new possibilities for developing group III metabotropic glutamate receptor agonists.

Selvam C, Oueslati N, Lemasson IA, Brabet I, Rigault D, Courtiol T, Cesarini S, Triballeau N, Bertrand HO, Goudet C, Pin JP, Acher FC. Selvam C, et al. Among authors: triballeau n. J Med Chem. 2010 Apr 8;53(7):2797-813. doi: 10.1021/jm901523t. J Med Chem. 2010. PMID: 20218620

2

Closure of the Venus flytrap module of mGlu8 receptor and the activation process: Insights from mutations converting antagonists into agonists.

Bessis AS, Rondard P, Gaven F, Brabet I, Triballeau N, Prezeau L, Acher F, Pin JP. Bessis AS, et al. Among authors: triballeau n. Proc Natl Acad Sci U S A. 2002 Aug 20;99(17):11097-102. doi: 10.1073/pnas.162138699. Epub 2002 Jul 31. Proc Natl Acad Sci U S A. 2002. PMID: 12151600 Free PMC article.

3

Virtual screening workflow development guided by the "receiver operating characteristic" curve approach. Application to high-throughput docking on metabotropic glutamate receptor subtype 4.

Triballeau N, Acher F, Brabet I, Pin JP, Bertrand HO. Triballeau N, et al. J Med Chem. 2005 Apr 7;48(7):2534-47. doi: 10.1021/jm049092j. J Med Chem. 2005. PMID: 15801843

4

Design and synthesis of APTCs (aminopyrrolidinetricarboxylic acids): identification of a new group III metabotropic glutamate receptor selective agonist.

Schann S, Menet C, Arvault P, Mercier G, Frauli M, Mayer S, Hubert N, Triballeau N, Bertrand HO, Acher F, Neuville P. Schann S, et al. Among authors: triballeau n. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4856-60. doi: 10.1016/j.bmcl.2006.06.062. Epub 2006 Jul 7. Bioorg Med Chem Lett. 2006. PMID: 16828551

5

High-potency olfactory receptor agonists discovered by virtual high-throughput screening: molecular probes for receptor structure and olfactory function.

Triballeau N, Van Name E, Laslier G, Cai D, Paillard G, Sorensen PW, Hoffmann R, Bertrand HO, Ngai J, Acher FC. Triballeau N, et al. Neuron. 2008 Dec 10;60(5):767-74. doi: 10.1016/j.neuron.2008.11.014. Neuron. 2008. PMID: 19081373 Free PMC article.

6

Identification of a novel NR2B-selective NMDA receptor antagonist using a virtual screening approach.

Mony L, Triballeau N, Paoletti P, Acher FC, Bertrand HO. Mony L, et al. Among authors: triballeau n. Bioorg Med Chem Lett. 2010 Sep 15;20(18):5552-8. doi: 10.1016/j.bmcl.2010.07.043. Epub 2010 Jul 15. Bioorg Med Chem Lett. 2010. PMID: 20692832

7

Rose Bengal analogs and vesicular glutamate transporters (VGLUTs).

Pietrancosta N, Kessler A, Favre-Besse FC, Triballeau N, Quentin T, Giros B, El Mestikawy S, Acher FC. Pietrancosta N, et al. Among authors: triballeau n. Bioorg Med Chem. 2010 Sep 15;18(18):6922-33. doi: 10.1016/j.bmc.2010.06.069. Epub 2010 Jun 25. Bioorg Med Chem. 2010. PMID: 20708942

8

Amino-pyrrolidine tricarboxylic acids give new insight into group III metabotropic glutamate receptor activation mechanism.

Frauli M, Hubert N, Schann S, Triballeau N, Bertrand HO, Acher F, Neuville P, Pin JP, Prézeau L. Frauli M, et al. Among authors: triballeau n. Mol Pharmacol. 2007 Mar;71(3):704-12. doi: 10.1124/mol.106.030254. Epub 2006 Dec 13. Mol Pharmacol. 2007. PMID: 17167031

9

Discovery of diarylhydantoins as new selective androgen receptor modulators.

Nique F, Hebbe S, Peixoto C, Annoot D, Lefrançois JM, Duval E, Michoux L, Triballeau N, Lemoullec JM, Mollat P, Thauvin M, Prangé T, Minet D, Clément-Lacroix P, Robin-Jagerschmidt C, Fleury D, Guédin D, Deprez P. Nique F, et al. Among authors: triballeau n. J Med Chem. 2012 Oct 11;55(19):8225-35. doi: 10.1021/jm300249m. Epub 2012 Sep 25. J Med Chem. 2012. PMID: 22897611

10

Discovery and optimization of an azetidine chemical series as a free fatty acid receptor 2 (FFA2) antagonist: from hit to clinic.

Pizzonero M, Dupont S, Babel M, Beaumont S, Bienvenu N, Blanqué R, Cherel L, Christophe T, Crescenzi B, De Lemos E, Delerive P, Deprez P, De Vos S, Djata F, Fletcher S, Kopiejewski S, L'Ebraly C, Lefrançois JM, Lavazais S, Manioc M, Nelles L, Oste L, Polancec D, Quénéhen V, Soulas F, Triballeau N, van der Aar EM, Vandeghinste N, Wakselman E, Brys R, Saniere L. Pizzonero M, et al. Among authors: triballeau n. J Med Chem. 2014 Dec 11;57(23):10044-57. doi: 10.1021/jm5012885. Epub 2014 Dec 1. J Med Chem. 2014. PMID: 25380412

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