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Page 1
Design, synthesis and efficacy of novel G protein-coupled receptor kinase 2 inhibitors.
Carotenuto A, Cipolletta E, Gomez-Monterrey I, Sala M, Vernieri E, Limatola A, Bertamino A, Musella S, Sorriento D, Grieco P, Trimarco B, Novellino E, Iaccarino G, Campiglia P. Carotenuto A, et al. Among authors: vernieri e. Eur J Med Chem. 2013 Nov;69:384-92. doi: 10.1016/j.ejmech.2013.08.039. Epub 2013 Sep 13. Eur J Med Chem. 2013. PMID: 24077529
Characterization of a selective CaMKII peptide inhibitor.
Gomez-Monterrey I, Sala M, Rusciano MR, Monaco S, Maione AS, Iaccarino G, Tortorella P, D'Ursi AM, Scrima M, Carotenuto A, De Rosa G, Bertamino A, Vernieri E, Grieco P, Novellino E, Illario M, Campiglia P. Gomez-Monterrey I, et al. Among authors: vernieri e. Eur J Med Chem. 2013 Apr;62:425-34. doi: 10.1016/j.ejmech.2012.12.053. Epub 2013 Jan 22. Eur J Med Chem. 2013. PMID: 23395965
Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors.
Vernieri E, Gomez-Monterrey I, Milite C, Grieco P, Musella S, Bertamino A, Scognamiglio I, Alcaro S, Artese A, Ortuso F, Novellino E, Sala M, Campiglia P. Vernieri E, et al. J Amino Acids. 2013;2013:606282. doi: 10.1155/2013/606282. Epub 2013 Feb 26. J Amino Acids. 2013. PMID: 23533709 Free PMC article.
Amino Acid derivatives as new zinc binding groups for the design of selective matrix metalloproteinase inhibitors.
Giustiniano M, Tortorella P, Agamennone M, Di Pizio A, Rossello A, Nuti E, Gomez-Monterrey I, Novellino E, Campiglia P, Vernieri E, Sala M, Bertamino A, Carotenuto A. Giustiniano M, et al. Among authors: vernieri e. J Amino Acids. 2013;2013:178381. doi: 10.1155/2013/178381. Epub 2013 Mar 10. J Amino Acids. 2013. PMID: 23555050 Free PMC article.
Discovery of PTPRJ agonist peptides that effectively inhibit in vitro cancer cell proliferation and tube formation.
Ortuso F, Paduano F, Carotenuto A, Gomez-Monterrey I, Bilotta A, Gaudio E, Sala M, Artese A, Vernieri E, Dattilo V, Iuliano R, Brancaccio D, Bertamino A, Musella S, Alcaro S, Grieco P, Perrotti N, Croce CM, Novellino E, Fusco A, Campiglia P, Trapasso F. Ortuso F, et al. Among authors: vernieri e. ACS Chem Biol. 2013 Jul 19;8(7):1497-506. doi: 10.1021/cb3007192. Epub 2013 May 13. ACS Chem Biol. 2013. PMID: 23627474
Synthesis, in vitro, and in cell studies of a new series of [indoline-3,2'-thiazolidine]-based p53 modulators.
Bertamino A, Soprano M, Musella S, Rusciano MR, Sala M, Vernieri E, Di Sarno V, Limatola A, Carotenuto A, Cosconati S, Grieco P, Novellino E, Illario M, Campiglia P, Gomez-Monterrey I. Bertamino A, et al. Among authors: vernieri e. J Med Chem. 2013 Jul 11;56(13):5407-21. doi: 10.1021/jm400311n. Epub 2013 Jun 26. J Med Chem. 2013. PMID: 23802716
Development and Identification of a Novel Anti-HIV-1 Peptide Derived by Modification of the N-Terminal Domain of HIV-1 Integrase.
Sala M, Spensiero A, Esposito F, Scala MC, Vernieri E, Bertamino A, Manfra M, Carotenuto A, Grieco P, Novellino E, Cadeddu M, Tramontano E, Schols D, Campiglia P, Gomez-Monterrey IM. Sala M, et al. Among authors: vernieri e. Front Microbiol. 2016 Jun 10;7:845. doi: 10.3389/fmicb.2016.00845. eCollection 2016. Front Microbiol. 2016. PMID: 27375570 Free PMC article.
An optimized Fmoc synthesis of human defensin 5.
Vernieri E, Valle J, Andreu D, de la Torre BG. Vernieri E, et al. Amino Acids. 2014 Feb;46(2):395-400. doi: 10.1007/s00726-013-1629-3. Epub 2013 Dec 6. Amino Acids. 2014. PMID: 24311274