BLU-451, a CNS-Active, Potent, and Selective Small-Molecule Inhibitor Against Uncommon EGFR Mutations.
Millet YA, Spira AI, Baik CS, Hong MH, Shum E, Patel JD, Nguyen D, Janne PA, Piotrowska Z, Leighl NB, Matsumoto S, Sun L, Yang TY, Yoshida T, Nilsson MB, Heymach JV, Murray BW, Keats J, Lee S, Hsieh J, Zalutskaya A, Le X.
Millet YA, et al. Among authors: yang ty.
Mol Cancer Ther. 2026 May 13. doi: 10.1158/1535-7163.MCT-25-1056. Online ahead of print.
Mol Cancer Ther. 2026.
PMID: 42126003