Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
7 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Pyrimidine derivatives as potent and selective A3 adenosine receptor antagonists.
J Med Chem. 2011 Jan 27;54(2):457-71. doi: 10.1021/jm100843z. Epub 2010 Dec 27.
J Med Chem. 2011.
PMID: 21186795
Divergent solution-phase synthesis of diarylpyrimidine libraries as selective A3 adenosine receptor antagonists.
Yaziji V, Coelho A, El Maatougui A, Brea J, Loza MI, Garcia-Mera X, Sotelo E.
Yaziji V, et al.
J Comb Chem. 2009 Jul-Aug;11(4):519-22. doi: 10.1021/cc900044k.
J Comb Chem. 2009.
PMID: 19472983
Item in Clipboard
Selective and potent adenosine A3 receptor antagonists by methoxyaryl substitution on the N-(2,6-diarylpyrimidin-4-yl)acetamide scaffold.
Yaziji V, Rodríguez D, Coelho A, García-Mera X, El Maatougui A, Brea J, Loza MI, Cadavid MI, Gutiérrez-de-Terán H, Sotelo E.
Yaziji V, et al.
Eur J Med Chem. 2013 Jan;59:235-42. doi: 10.1016/j.ejmech.2012.11.010. Epub 2012 Nov 24.
Eur J Med Chem. 2013.
PMID: 23231967
Item in Clipboard
Effect of Nitrogen Atom Substitution in A3 Adenosine Receptor Binding: N-(4,6-Diarylpyridin-2-yl)acetamides as Potent and Selective Antagonists.
Azuaje J, Jespers W, Yaziji V, Mallo A, Majellaro M, Caamaño O, Loza MI, Cadavid MI, Brea J, Åqvist J, Sotelo E, Gutiérrez-de-Terán H.
Azuaje J, et al. Among authors: yaziji v.
J Med Chem. 2017 Sep 14;60(17):7502-7511. doi: 10.1021/acs.jmedchem.7b00860. Epub 2017 Aug 21.
J Med Chem. 2017.
PMID: 28792759
Item in Clipboard
Discovery and preliminary SAR of 5-arylidene-2,2-dimethyl-1,3-dioxane- 4,6-diones as platelet aggregation inhibitors.
El Maatougui A, Azuaje J, Coelho A, Cano E, Yañez M, López C, Yaziji V, Carbajales C, Sotelo E.
El Maatougui A, et al. Among authors: yaziji v.
Comb Chem High Throughput Screen. 2012 Aug;15(7):551-4. doi: 10.2174/138620712801619122.
Comb Chem High Throughput Screen. 2012.
PMID: 22272691
Item in Clipboard
Three-component assembly of structurally diverse 2-aminopyrimidine-5-carbonitriles.
Val C, Crespo A, Yaziji V, Coelho A, Azuaje J, El Maatougui A, Carbajales C, Sotelo E.
Val C, et al. Among authors: yaziji v.
ACS Comb Sci. 2013 Jul 8;15(7):370-8. doi: 10.1021/co4000503. Epub 2013 Jun 6.
ACS Comb Sci. 2013.
PMID: 23697392
Item in Clipboard
Integrated Ugi-based assembly of functionally, skeletally, and stereochemically diverse 1,4-benzodiazepin-2-ones.
Azuaje J, Pérez-Rubio JM, Yaziji V, El Maatougui A, González-Gomez JC, Sánchez-Pedregal VM, Navarro-Vázquez A, Masaguer CF, Teijeira M, Sotelo E.
Azuaje J, et al. Among authors: yaziji v.
J Org Chem. 2015 Feb 6;80(3):1533-49. doi: 10.1021/jo502382q. Epub 2015 Jan 20.
J Org Chem. 2015.
PMID: 25560990
Free article.
Item in Clipboard
Cite
Cite