The zymogenic form of SARS-CoV-2 main protease: A discrete target for drug discovery.
Novotný P, Humpolíčková J, Nováková V, Stanchev S, Stříšovský K, Zgarbová M, Weber J, Kryštůfek R, Starková J, Hradilek M, Moravcová A, Günterová J, Bach K, Majer P, Konvalinka J, Majerová T.
Novotný P, et al.
J Biol Chem. 2024 Dec 14;301(1):108079. doi: 10.1016/j.jbc.2024.108079. Online ahead of print.
J Biol Chem. 2024.
PMID: 39675720
Free article.
Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) main protease (M(pro)) autocatalytically releases itself out of the viral polyprotein to form a fully active mature dimer in a manner that is not fully understood. ...Our findings help expand unders …
Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) main protease (M(pro)) autocatalytically releases itself o …