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Table representation of search results timeline featuring number of search results per year.

Year Number of Results
2001 2
2002 4
2003 2
2004 3
2005 3
2006 1
2007 1
2008 3
2009 2
2010 1
2011 2
2012 2
2013 6
2014 2
2015 4
2016 10
2017 7
2018 8
2019 3
2020 7
2021 6
2022 6
2023 9
2024 4
2025 9
2026 1

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100 results

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Page 1
Development of Biphenyl-Substituted Uracil-Based Hydroxamic Acids (UBHAs) as Potent HDAC Inhibitors with Pro-Apoptotic Activity in Leukemia and Prostate Cancer Cells.
Fiorentino F, Bontempi G, Michetti F, Pecci V, Fabbrizi E, Passeri D, Corsetti L, Farini V, Casano F, Gioiello A, Di Sotto A, Pellicciari R, Bufalo DD, Trisciuoglio D, Nanni S, Strippoli R, Mai A, Rotili D. Fiorentino F, et al. Among authors: trisciuoglio d. J Med Chem. 2026 May 14;69(9):10060-10082. doi: 10.1021/acs.jmedchem.5c02737. Epub 2026 Apr 30. J Med Chem. 2026. PMID: 42059134 Free PMC article.
Quinoline-Based DNA Methyltransferase Inhibitors Featuring Basic Side Chains: Design, Synthesis, and Insight in Biochemical and Anticancer Cell Properties.
Zwergel C, Lambona C, Fioravanti R, Raucci A, Fiorentino F, Nchugoua Tchieh G, Jallet C, Lacroix L, Pierrettori M, Pellegrini FR, Xiong Y, Jin J, Arimondo P, Trisciuoglio D, Mai A, Valente S. Zwergel C, et al. Among authors: trisciuoglio d. J Med Chem. 2025 Nov 27;68(22):23886-23909. doi: 10.1021/acs.jmedchem.5c01029. Epub 2025 Nov 11. J Med Chem. 2025. PMID: 41217771 Free PMC article.
Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells.
Bozdag M, Mroweh N, Raucci A, Angeli A, Peppicelli S, Biagioni A, Calorini L, Trisciuoglio D, Ragno R, Astolfi R, Giuliani L, Zwergel C, Valente S, Andreucci E, Carta F, Mai A, Supuran CT. Bozdag M, et al. Among authors: trisciuoglio d. J Med Chem. 2025 Nov 13;68(21):22874-22895. doi: 10.1021/acs.jmedchem.5c01788. Epub 2025 Oct 28. J Med Chem. 2025. PMID: 41150938 Free PMC article.
Reverse transcriptase inhibitors induce autophagy in a LINE-1 ORF1p-dependent manner.
Damizia M, Baranzini M, Sciamanna I, Altieri L, Rovella P, Rosas Bringa OG, Hozeifi S, Saba LJ, Mourtzinos A, O'Shea A, Ansari MSZ, Andreola F, Cirilli R, Sbardella G, Serafino A, Schumann GG, Trisciuoglio D, LaCava J, Lavia P, Spadafora C. Damizia M, et al. Among authors: trisciuoglio d. bioRxiv [Preprint]. 2025 Aug 12:2025.08.07.669170. doi: 10.1101/2025.08.07.669170. bioRxiv. 2025. PMID: 40832305 Free PMC article. Preprint.
NF-κB-mediated cytokine secretion and glutamate metabolic reprogramming converge in breast cancer brain tropism.
Di Russo S, Borsatti GE, Bouzidi A, Liberati FR, Riva A, Tripodi F, Rolfi LR, Spizzichino S, Tramutola A, Perluigi M, Trisciuoglio D, Giardina G, Paiardini A, Coccetti P, Rinaldo S, Cutruzzolà F, Paone A. Di Russo S, et al. Among authors: trisciuoglio d. Cancer Lett. 2025 Oct 10;630:217907. doi: 10.1016/j.canlet.2025.217907. Epub 2025 Jul 8. Cancer Lett. 2025. PMID: 40639610 Free article.
Tranylcypromine-Based LSD1 Inhibitors as Useful Agents to Reduce Viability of Schistosoma mansoni.
Fabbrizi E, Hailu GS, Ganesan A, Fioravanti R, Zwergel C, Lambona C, Valente S, Fianco G, Iuzzolino A, Trisciuoglio D, Caroli J, Mattevi A, Häberli C, Keiser J, Rotili D, Mai A. Fabbrizi E, et al. Among authors: trisciuoglio d. ACS Infect Dis. 2025 Aug 8;11(8):2178-2189. doi: 10.1021/acsinfecdis.5c00224. Epub 2025 Jul 2. ACS Infect Dis. 2025. PMID: 40601861 Free PMC article.
Interplay between ALK2R206H mutant receptor and autophagy signaling regulates receptor stability and its chondrogenic functions.
Coculo L, Wits M, Mariani I, Fianco G, Cappato S, Bocciardi R, Pedemonte N, Volpe E, Ciolfi S, Sessa RL, Rinaldo S, Cutruzzolà F, Trisciuoglio D, Goumans MJ, Sanchez-Duffhues G, Stagni V. Coculo L, et al. Among authors: trisciuoglio d. Cell Death Discov. 2025 Mar 22;11(1):117. doi: 10.1038/s41420-025-02393-0. Cell Death Discov. 2025. PMID: 40121219 Free PMC article.
100 results