Reg2 inactivation increases sensitivity to Fas hepatotoxicity and delays liver regeneration post-hepatectomy in mice

Hepatology. 2006 Dec;44(6):1452-64. doi: 10.1002/hep.21434.

Abstract

Reg2/RegIIIbeta is the murine homologue of the human secreted HIP/PAP C-type lectin. HIP/PAP transgenic mice were protected against acetaminophen-induced acute liver failure and were stimulated to regenerate post-hepatectomy. To assess the role of Reg2, we used Reg2-/- mice in a model of fulminant hepatitis induced by Fas and in the post-hepatectomy regeneration. Within 4 hours of J0-2 treatment (0.5 microg/g), only 50% of the Reg2-/- mice were alive but with an increased sensitivity to Fas-induced oxidative stress and a decreased level of Bcl-xL. In contrast, HIP/PAP transgenic mice were resistant to Fas, with HIP/PAP serving as a sulfhydryl buffer to slow down decreases in glutathione and Bcl-xL. In Reg2-/- mice, liver regeneration was markedly impaired, with 29% mortality and delay of the S-phase and the activation of ERK1/2 and AKT. Activation of STAT3 began on time at 3 hours but persisted strongly up to 72 hours despite significant accumulation of SOCS3. Thus, Reg2 deficiency induced exaggerated IL-6/STAT-3 activation and mito-inhibition. Because the Reg2 gene was activated between 6 and 24 hours after hepatectomy in wild-type mice, Reg2 could mediate the TNF-alpha/IL-6 priming signaling by exerting a negative feed-back on STAT3/IL-6 activation to allow the hepatocytes to progress through the cell cycle. In conclusion, Reg2 deficiency enhanced liver sensitivity to Fas-induced oxidative stress and delayed liver regeneration with persistent TNF-alpha/IL6/STAT3 signaling. In contrast, overexpression of human HIP/PAP promoted liver resistance to Fas and accelerated liver regeneration with early activation/deactivation of STAT3. Reg2/HIP/PAP is therefore a critical mitogenic and antiapoptotic factor for the liver.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibodies, Monoclonal
  • Antigens, Neoplasm / physiology
  • Biomarkers, Tumor / physiology
  • Chemical and Drug Induced Liver Injury
  • DNA / biosynthesis
  • Extracellular Signal-Regulated MAP Kinases / metabolism
  • Hepatectomy
  • Humans
  • Hydrazines
  • Interleukin-6 / physiology
  • Lectins, C-Type / physiology
  • Liver Regeneration / physiology*
  • Mice
  • Mice, Transgenic
  • Oncogene Protein v-akt / physiology
  • Pancreatitis-Associated Proteins
  • Proteins / physiology*
  • Pyrazines
  • Quinolines
  • Signal Transduction / physiology
  • Tumor Necrosis Factor-alpha / physiology
  • fas Receptor / physiology*

Substances

  • Antibodies, Monoclonal
  • Antigens, Neoplasm
  • Biomarkers, Tumor
  • Fas protein, mouse
  • Hydrazines
  • Interleukin-6
  • Lectins, C-Type
  • Pancreatitis-Associated Proteins
  • Proteins
  • Pyrazines
  • QU663 compound
  • Quinolines
  • REG3A protein, human
  • Reg3b protein, mouse
  • Tumor Necrosis Factor-alpha
  • fas Receptor
  • DNA
  • Oncogene Protein v-akt
  • Extracellular Signal-Regulated MAP Kinases