Effects of a CRF2R agonist and exercise on mdx and wildtype skeletal muscle

Muscle Nerve. 2007 Sep;36(3):336-41. doi: 10.1002/mus.20820.

Abstract

Corticotrophin-releasing factor 2 receptor (CRF2R) agonists prevent muscle atrophy due to immobilization, denervation, and corticosteroid-induced muscle atrophy in wildtype mice. We hypothesized that a CRF2R agonist will increase skeletal muscle mass in mdx mice. Mdx (C57BL/10ScSn-Dmd(mdx)) and wildtype (C57BL/6) mice were divided into four groups: sedentary placebo, sedentary CRF2R agonist, exercised placebo, and exercised CRF2R agonist. Mice exercised on a treadmill twice weekly for 30 min (8-12 m/min, 8 weeks). Muscle and heart weights, serum creatine kinase, and gamma-glutamyltransferase activities were measured. The CRF2R agonist increased extensor digitorum longus and soleus muscle weights (P < 0.05) in wildtype and mdx mice. Sedentary mdx CRF2R and exercised mdx placebo mice had lower serum creatine kinase activity than sedentary mdx placebo mice. CRF2R-treated mice had decreased heart weights compared to placebo-treated mice. We conclude that CRF2R agonists should be further evaluated as a potential therapy for dystrophinopathies.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Body Weight
  • Creatine Kinase / blood
  • Heart / anatomy & histology
  • Mice
  • Mice, Inbred C57BL
  • Mice, Inbred mdx
  • Muscle, Skeletal / anatomy & histology
  • Muscle, Skeletal / chemistry
  • Muscle, Skeletal / drug effects*
  • Organ Size
  • Physical Conditioning, Animal
  • Proteins / analysis
  • Receptors, Corticotropin-Releasing Hormone / agonists*
  • gamma-Glutamyltransferase / blood

Substances

  • CRF receptor type 2
  • Proteins
  • Receptors, Corticotropin-Releasing Hormone
  • gamma-Glutamyltransferase
  • Creatine Kinase