Strain-promoted copper-free "click" chemistry for 18F radiolabeling of bombesin

Angew Chem Int Ed Engl. 2011 Nov 18;50(47):11117-20. doi: 10.1002/anie.201105547. Epub 2011 Sep 28.
No abstract available

MeSH terms

  • Azides / chemistry
  • Binding, Competitive
  • Bombesin / analogs & derivatives*
  • Bombesin / chemical synthesis
  • Bombesin / chemistry
  • Cell Line, Tumor
  • Click Chemistry / methods*
  • Copper / chemistry
  • Fluorine Radioisotopes
  • Humans
  • Isotope Labeling
  • Molecular Structure
  • Positron-Emission Tomography
  • Protein Binding
  • Radioligand Assay
  • Radiopharmaceuticals / chemical synthesis*
  • Radiopharmaceuticals / chemistry
  • Receptors, Bombesin / antagonists & inhibitors
  • Receptors, Bombesin / metabolism

Substances

  • Azides
  • Fluorine Radioisotopes
  • Radiopharmaceuticals
  • Receptors, Bombesin
  • bombesin, Lys(3)-
  • Copper
  • Bombesin