Abstract
The affinity of LY-171555 (quinpirole) and BHT-920 for both states of rat striatal dopamine D-1 and D-2 receptors was determined. Although these drugs have different pharmacological effects in experimental animals, we found that they had similar affinities for both D-1 and D-2 receptors.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Animals
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Azepines / metabolism*
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Benzazepines / pharmacology
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Corpus Striatum / metabolism*
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Dopamine Agents / metabolism*
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Endothelins
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Ergolines / metabolism*
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Guanylyl Imidodiphosphate / pharmacology
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In Vitro Techniques
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Male
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Peptides / pharmacology*
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Quinpirole
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Rats
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Rats, Inbred Strains
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Receptors, Dopamine / metabolism*
Substances
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Azepines
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Benzazepines
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Dopamine Agents
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Endothelins
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Ergolines
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Peptides
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Receptors, Dopamine
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Quinpirole
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Guanylyl Imidodiphosphate
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talipexole