Small molecules and their role in effective preclinical target validation

Future Med Chem. 2017 Sep;9(14):1579-1582. doi: 10.4155/fmc-2017-0121. Epub 2017 Aug 22.
No abstract available

Keywords: bromodomain; chemical probe; target validation.

Publication types

  • Editorial

MeSH terms

  • Drug Discovery / methods*
  • Drug Discovery / standards
  • Humans
  • Molecular Probes / chemistry
  • Molecular Probes / pharmacology*
  • Molecular Targeted Therapy / methods*
  • Molecular Targeted Therapy / standards
  • Pharmaceutical Preparations / chemistry*
  • Reproducibility of Results
  • Small Molecule Libraries / chemistry
  • Small Molecule Libraries / pharmacology*

Substances

  • Molecular Probes
  • Pharmaceutical Preparations
  • Small Molecule Libraries