Isolation and characterization of ARA160 as the first androgen receptor N-terminal-associated coactivator in human prostate cells

J Biol Chem. 1999 Aug 6;274(32):22373-9. doi: 10.1074/jbc.274.32.22373.

Abstract

The androgen receptor (AR) is a member of the steroid receptor superfamily that may require coactivators for proper or maximal transactivation. Using a purified AR N-terminal peptide as a probe to screen the human testis expression library, we identified an androgen-enhanced AR N-terminal-associated protein ARA160, which consists of 1,093 amino acids with an apparent molecular mass of 160 kDa. Sequence comparison in GenBank(TM) reveals that ARA160 shares an identical sequence with a HIV-1 TATA element modulatory factor, TMF. The far-Western blotting and co-immunoprecipitation assays demonstrate that the AR can interact directly with ARA160/TMF. Affinity gel pull-down and mammalian two-hybrid assays further suggest androgen can enhance significantly the interaction between AR and ARA160. Transient transfection assays demonstrated that ARA160 might function as a coactivator for AR-mediated transactivation in human prostate cancer PC-3 cells. Our data further suggest that this AR N-terminal coactivator can function cooperatively with AR C-terminal coactivator, ARA70, in PC-3 cells. Together, our data demonstrate that ARA160 might represent the first identified androgen-enhanced N-terminal coactivator for the AR.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Androgens / metabolism*
  • Cloning, Molecular
  • DNA-Binding Proteins / genetics
  • DNA-Binding Proteins / isolation & purification
  • DNA-Binding Proteins / metabolism*
  • Humans
  • Ligands
  • Male
  • Mammary Tumor Virus, Mouse / genetics
  • Molecular Sequence Data
  • Nuclear Receptor Coactivators
  • Oncogene Proteins*
  • Promoter Regions, Genetic
  • Prostate / chemistry
  • Prostate / metabolism*
  • Prostate-Specific Antigen / genetics
  • Protein Binding
  • Receptors, Androgen / metabolism*
  • Receptors, Estrogen / metabolism
  • Receptors, Glucocorticoid / metabolism
  • Response Elements
  • Sequence Analysis, DNA
  • Terminal Repeat Sequences
  • Trans-Activators / metabolism
  • Transcription Factors / genetics
  • Transcription Factors / isolation & purification
  • Transcription Factors / metabolism*
  • Transcriptional Activation

Substances

  • Androgens
  • DNA-Binding Proteins
  • Ligands
  • NCOA4 protein, human
  • Nuclear Receptor Coactivators
  • Oncogene Proteins
  • Receptors, Androgen
  • Receptors, Estrogen
  • Receptors, Glucocorticoid
  • Trans-Activators
  • Transcription Factors
  • TMF1 protein, human
  • Prostate-Specific Antigen