Potent neutralization of botulinum neurotoxin by recombinant oligoclonal antibody

Proc Natl Acad Sci U S A. 2002 Aug 20;99(17):11346-50. doi: 10.1073/pnas.172229899. Epub 2002 Aug 12.

Abstract

The botulinum neurotoxins (BoNTs) cause the paralytic human disease botulism and are one of the highest-risk threat agents for bioterrorism. To generate a pharmaceutical to prevent or treat botulism, monoclonal antibodies (mAbs) were generated by phage display and evaluated for neutralization of BoNT serotype A (BoNT/A) in vivo. Although no single mAb significantly neutralized toxin, a combination of three mAbs (oligoclonal Ab) neutralized 450,000 50% lethal doses of BoNT/A, a potency 90 times greater than human hyperimmune globulin. The potency of oligoclonal Ab was primarily due to a large increase in functional Ab binding affinity. The results indicate that the potency of the polyclonal humoral immune response can be deconvoluted to a few mAbs binding nonoverlapping epitopes, providing a route to drugs for preventing and treating botulism and diseases caused by other pathogens and biologic threat agents.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Antibodies, Bacterial / immunology*
  • Antibodies, Monoclonal / immunology*
  • Antibody Specificity
  • Base Sequence
  • Botulinum Toxins / immunology*
  • DNA Primers
  • Immunoglobulin G / immunology*
  • Immunoglobulin Heavy Chains / genetics
  • Immunoglobulin Heavy Chains / immunology
  • Kinetics
  • Male
  • Mice
  • Neutralization Tests
  • Phrenic Nerve / immunology
  • Polymerase Chain Reaction
  • Recombinant Proteins / immunology
  • Time Factors

Substances

  • Antibodies, Bacterial
  • Antibodies, Monoclonal
  • DNA Primers
  • Immunoglobulin G
  • Immunoglobulin Heavy Chains
  • Recombinant Proteins
  • Botulinum Toxins