Effects of Cordyceps militaris extract on angiogenesis and tumor growth

Acta Pharmacol Sin. 2004 May;25(5):657-65.

Abstract

Aim: To evaluate the effects of Cordyceps militaris extract (CME) on angiogenesis and tumor growth.

Methods: Human umbilical vein endothelial cells (HUVEC), HT1080, and B16-F10 cells were used. DNA fragment, angiogenic related gene expressions (MMPs, bFGF, VEGF, etc), capillary tube formation, wound healing in vitro, tumor growth in vivo were measured.

Results: CME inhibited growth of HUVECs and HT1080 (P<0.01). CME 100 and 200 mg/L reduced MMP-2 gene expression in HT1080 cells by 6.0 % and 22.9 % after 3-h and 14.9 % and 32.8 % after 6-h treatment. CME did not affect MMP-9 gene expression in B16-F10 melanoma cells. CME 100 and 200 mg/L also reduced bFGF gene expression in HUVECs by 22.2 % and 41.3 %. CME inhibited tube formation of endothelial cells in vitro and in vivo. CME repressed the growth of B16-F10 melanoma cells in mice compared with control group (P<0.05).

Conclusion: CME has antiangiogenetic properties.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Division / drug effects
  • Cells, Cultured
  • Cordyceps* / chemistry
  • Drugs, Chinese Herbal / isolation & purification
  • Drugs, Chinese Herbal / pharmacology*
  • Endothelial Cells / drug effects
  • Endothelial Cells / metabolism
  • Fibroblast Growth Factor 2 / biosynthesis*
  • Fibroblast Growth Factor 2 / genetics
  • Fibrosarcoma / pathology
  • Humans
  • Matrix Metalloproteinase 2 / biosynthesis
  • Matrix Metalloproteinase 2 / genetics
  • Matrix Metalloproteinase 9 / biosynthesis
  • Matrix Metalloproteinase 9 / genetics
  • Melanoma, Experimental / pathology*
  • Mice
  • Mice, Inbred C57BL
  • Neovascularization, Pathologic / metabolism*
  • Plants, Medicinal / chemistry
  • RNA, Messenger / genetics
  • Tumor Cells, Cultured
  • Umbilical Veins / cytology

Substances

  • Drugs, Chinese Herbal
  • RNA, Messenger
  • Fibroblast Growth Factor 2
  • Matrix Metalloproteinase 2
  • Matrix Metalloproteinase 9