Tebben AJ - Search Results

1

Capped diaminopropionamide-glycine dipeptides are inhibitors of CC chemokine receptor 2 (CCR2).

Carter PH, Brown GD, Friedrich SR, Cherney RJ, Tebben AJ, Lo YC, Yang G, Jezak H, Solomon KA, Scherle PA, Decicco CP. Carter PH, et al. Among authors: tebben aj. Bioorg Med Chem Lett. 2007 Oct 1;17(19):5455-61. doi: 10.1016/j.bmcl.2007.07.028. Epub 2007 Jul 21. Bioorg Med Chem Lett. 2007. PMID: 17720492

2

A molecular modeling analysis of novel non-hydroxamate inhibitors of TACE.

Sheppeck JE 2nd, Tebben A, Gilmore JL, Yang A, Wasserman ZR, Decicco CP, Duan JJ. Sheppeck JE 2nd, et al. Bioorg Med Chem Lett. 2007 Mar 1;17(5):1408-12. doi: 10.1016/j.bmcl.2006.11.082. Epub 2006 Dec 3. Bioorg Med Chem Lett. 2007. PMID: 17188861

3

Both 5-arylidene-2-thioxodihydropyrimidine-4,6(1H,5H)-diones and 3-thioxo-2,3-dihydro-1H-imidazo[1,5-a]indol-1-ones are light-dependent tumor necrosis factor-alpha antagonists.

Voss ME, Carter PH, Tebben AJ, Scherle PA, Brown GD, Thompson LA, Xu M, Lo YC, Yang G, Liu RQ, Strzemienski P, Everlof JG, Trzaskos JM, Decicco CP. Voss ME, et al. Among authors: tebben aj. Bioorg Med Chem Lett. 2003 Feb 10;13(3):533-8. doi: 10.1016/s0960-894x(02)00941-1. Bioorg Med Chem Lett. 2003. PMID: 12565966

4

From rigid cyclic templates to conformationally stabilized acyclic scaffolds. Part I: the discovery of CCR3 antagonist development candidate BMS-639623 with picomolar inhibition potency against eosinophil chemotaxis.

Santella JB 3rd, Gardner DS, Yao W, Shi C, Reddy P, Tebben AJ, DeLucca GV, Wacker DA, Watson PS, Welch PK, Wadman EA, Davies P, Solomon KA, Graden DM, Yeleswaram S, Mandlekar S, Kariv I, Decicco CP, Ko SS, Carter PH, Duncia JV. Santella JB 3rd, et al. Among authors: tebben aj. Bioorg Med Chem Lett. 2008 Jan 15;18(2):576-85. doi: 10.1016/j.bmcl.2007.11.067. Epub 2007 Nov 22. Bioorg Med Chem Lett. 2008. PMID: 18096386

5

From rigid cyclic templates to conformationally stabilized acyclic scaffolds. Part II: Acyclic replacements for the (3S)-3-benzylpiperidine in a series of potent CCR3 antagonists.

Gardner DS, Santella JB 3rd, Tebben AJ, Batt DG, Ko SS, Traeger SC, Welch PK, Wadman EA, Davies P, Carter PH, Duncia JV. Gardner DS, et al. Among authors: tebben aj. Bioorg Med Chem Lett. 2008 Jan 15;18(2):586-95. doi: 10.1016/j.bmcl.2007.11.087. Epub 2007 Nov 28. Bioorg Med Chem Lett. 2008. PMID: 18160284

6

Discovery of disubstituted cyclohexanes as a new class of CC chemokine receptor 2 antagonists.

Cherney RJ, Mo R, Meyer DT, Nelson DJ, Lo YC, Yang G, Scherle PA, Mandlekar S, Wasserman ZR, Jezak H, Solomon KA, Tebben AJ, Carter PH, Decicco CP. Cherney RJ, et al. Among authors: tebben aj. J Med Chem. 2008 Feb 28;51(4):721-4. doi: 10.1021/jm701488f. Epub 2008 Jan 31. J Med Chem. 2008. PMID: 18232650

7

Chapter 12. The use of receptor homology modeling to facilitate the design of selective chemokine receptor antagonists.

Carter PH, Tebben AJ. Carter PH, et al. Among authors: tebben aj. Methods Enzymol. 2009;461:249-79. doi: 10.1016/S0076-6879(09)05412-3. Methods Enzymol. 2009. PMID: 19480923

8

Novel sulfone-containing di- and trisubstituted cyclohexanes as potent CC chemokine receptor 2 (CCR2) antagonists.

Cherney RJ, Mo R, Meyer DT, Voss ME, Lo YC, Yang G, Miller PB, Scherle PA, Tebben AJ, Carter PH, Decicco CP. Cherney RJ, et al. Among authors: tebben aj. Bioorg Med Chem Lett. 2009 Jul 1;19(13):3418-22. doi: 10.1016/j.bmcl.2009.05.041. Epub 2009 May 18. Bioorg Med Chem Lett. 2009. PMID: 19481449

9

Synthesis of 3-phenylsulfonylmethyl cyclohexylaminobenzamide-derived antagonists of CC chemokine receptor 2 (CCR2).

Yang MG, Xiao Z, Shi Q, Cherney RJ, Tebben AJ, De Lucca GV, Santella JB 3rd, Mo R, Cvijic ME, Zhao Q, Barrish JC, Carter PH. Yang MG, et al. Among authors: tebben aj. Bioorg Med Chem Lett. 2012 Feb 1;22(3):1384-7. doi: 10.1016/j.bmcl.2011.12.057. Epub 2011 Dec 16. Bioorg Med Chem Lett. 2012. PMID: 22225639

10

Discovery of an orally-bioavailable CC Chemokine Receptor 2 antagonist derived from an acyclic diaminoalcohol backbone.

Carter PH, Brown GD, King SR, Voss ME, Tebben AJ, Cherney RJ, Mandlekar S, Lo YC, Yang G, Miller PB, Scherle PA, Zhao Q, Decicco CP. Carter PH, et al. Among authors: tebben aj. Bioorg Med Chem Lett. 2012 May 1;22(9):3311-6. doi: 10.1016/j.bmcl.2012.03.007. Epub 2012 Mar 10. Bioorg Med Chem Lett. 2012. PMID: 22475558

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