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Exploring functional genomics for drug target and therapeutics discovery in Plasmodia.
Acta Trop. 2008 Feb;105(2):113-23. doi: 10.1016/j.actatropica.2007.10.013. Epub 2007 Nov 12.
Acta Trop. 2008.
PMID: 18083131
Review.
Functional consequences of perturbing polyamine metabolism in the malaria parasite, Plasmodium falciparum.
Clark K, Niemand J, Reeksting S, Smit S, van Brummelen AC, Williams M, Louw AI, Birkholtz L.
Clark K, et al. Among authors: van brummelen ac.
Amino Acids. 2010 Feb;38(2):633-44. doi: 10.1007/s00726-009-0424-7. Epub 2009 Dec 9.
Amino Acids. 2010.
PMID: 19997948
Review.
Item in Clipboard
Co-inhibition of Plasmodium falciparum S-adenosylmethionine decarboxylase/ornithine decarboxylase reveals perturbation-specific compensatory mechanisms by transcriptome, proteome, and metabolome analyses.
van Brummelen AC, Olszewski KL, Wilinski D, Llinás M, Louw AI, Birkholtz LM.
van Brummelen AC, et al.
J Biol Chem. 2009 Feb 13;284(7):4635-46. doi: 10.1074/jbc.M807085200. Epub 2008 Dec 10.
J Biol Chem. 2009.
PMID: 19073607
Free PMC article.
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Plasmodium falciparum spermidine synthase inhibition results in unique perturbation-specific effects observed on transcript, protein and metabolite levels.
Becker JV, Mtwisha L, Crampton BG, Stoychev S, van Brummelen AC, Reeksting S, Louw AI, Birkholtz LM, Mancama DT.
Becker JV, et al. Among authors: van brummelen ac.
BMC Genomics. 2010 Apr 12;11:235. doi: 10.1186/1471-2164-11-235.
BMC Genomics. 2010.
PMID: 20385001
Free PMC article.
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In vitro anti-plasmodial activity of Dicoma anomala subsp. gerrardii (Asteraceae): identification of its main active constituent, structure-activity relationship studies and gene expression profiling.
Becker JV, van der Merwe MM, van Brummelen AC, Pillay P, Crampton BG, Mmutlane EM, Parkinson C, van Heerden FR, Crouch NR, Smith PJ, Mancama DT, Maharaj VJ.
Becker JV, et al. Among authors: van brummelen ac.
Malar J. 2011 Oct 11;10:295. doi: 10.1186/1475-2875-10-295.
Malar J. 2011.
PMID: 21985233
Free PMC article.
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ATP and luciferase assays to determine the rate of drug action in in vitro cultures of Plasmodium falciparum.
Khan T, van Brummelen AC, Parkinson CJ, Hoppe HC.
Khan T, et al. Among authors: van brummelen ac.
Malar J. 2012 Nov 7;11:369. doi: 10.1186/1475-2875-11-369.
Malar J. 2012.
PMID: 23134617
Free PMC article.
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The potential role of resveratrol as supportive antiviral in treating conditions such as COVID-19 - A formulator's perspective.
van Brummelen R, van Brummelen AC.
van Brummelen R, et al. Among authors: van brummelen ac.
Biomed Pharmacother. 2022 Apr;148:112767. doi: 10.1016/j.biopha.2022.112767. Epub 2022 Feb 28.
Biomed Pharmacother. 2022.
PMID: 35240527
Free PMC article.
Review.
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