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Non-acidic pyrazole EP1 receptor antagonists with in vivo analgesic efficacy.
Bioorg Med Chem Lett. 2008 Jun 1;18(11):3392-9. doi: 10.1016/j.bmcl.2008.04.018. Epub 2008 Apr 11.
Bioorg Med Chem Lett. 2008.
PMID: 18462938
1,5-Biaryl pyrrole derivatives as EP1 receptor antagonists. Structure-activity relationships of 6-substituted and 5,6-disubstituted benzoic acid derivatives.
Hall A, Brown SH, Chessell IP, Chowdhury A, Clayton NM, Coleman T, Giblin GM, Hammond B, Healy MP, Johnson MR, Metcalf A, Michel AD, Naylor A, Novelli R, Spalding DJ, Sweeting J, Winyard L.
Hall A, et al. Among authors: winyard l.
Bioorg Med Chem Lett. 2007 Feb 15;17(4):916-20. doi: 10.1016/j.bmcl.2006.11.059. Epub 2006 Nov 22.
Bioorg Med Chem Lett. 2007.
PMID: 17175160
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An animal model of chronic inflammatory pain: pharmacological and temporal differentiation from acute models.
Wilson AW, Medhurst SJ, Dixon CI, Bontoft NC, Winyard LA, Brackenborough KT, De Alba J, Clarke CJ, Gunthorpe MJ, Hicks GA, Bountra C, McQueen DS, Chessell IP.
Wilson AW, et al. Among authors: winyard la.
Eur J Pain. 2006 Aug;10(6):537-49. doi: 10.1016/j.ejpain.2005.08.003. Epub 2005 Sep 30.
Eur J Pain. 2006.
PMID: 16199187
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Activation of CB1 and CB2 receptors attenuates the induction and maintenance of inflammatory pain in the rat.
Elmes SJR, Winyard LA, Medhurst SJ, Clayton NM, Wilson AW, Kendall DA, Chapman V.
Elmes SJR, et al. Among authors: winyard la.
Pain. 2005 Dec 5;118(3):327-335. doi: 10.1016/j.pain.2005.09.005. Epub 2005 Nov 14.
Pain. 2005.
PMID: 16289798
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Evaluation of the effects of lamotrigine, valproate and carbamazepine in a rodent model of mania.
Arban R, Maraia G, Brackenborough K, Winyard L, Wilson A, Gerrard P, Large C.
Arban R, et al. Among authors: winyard l.
Behav Brain Res. 2005 Mar 7;158(1):123-32. doi: 10.1016/j.bbr.2004.08.015.
Behav Brain Res. 2005.
PMID: 15680200
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