Zimmermann H - Search Results

1

Development of potent and selective inhibitors of ecto-5'-nucleotidase based on an anthraquinone scaffold.

Baqi Y, Lee SY, Iqbal J, Ripphausen P, Lehr A, Scheiff AB, Zimmermann H, Bajorath J, Müller CE. Baqi Y, et al. Among authors: zimmermann h. J Med Chem. 2010 Mar 11;53(5):2076-86. doi: 10.1021/jm901851t. J Med Chem. 2010. PMID: 20146483

2

Nucleoside-5'-monophosphates as prodrugs of adenosine A2A receptor agonists activated by ecto-5'-nucleotidase.

El-Tayeb A, Iqbal J, Behrenswerth A, Romio M, Schneider M, Zimmermann H, Schrader J, Müller CE. El-Tayeb A, et al. Among authors: zimmermann h. J Med Chem. 2009 Dec 10;52(23):7669-77. doi: 10.1021/jm900538v. J Med Chem. 2009. PMID: 19580286

3

Virtual screening identifies novel sulfonamide inhibitors of ecto-5'-nucleotidase.

Ripphausen P, Freundlieb M, Brunschweiger A, Zimmermann H, Müller CE, Bajorath J. Ripphausen P, et al. Among authors: zimmermann h. J Med Chem. 2012 Jul 26;55(14):6576-81. doi: 10.1021/jm300658n. Epub 2012 Jul 9. J Med Chem. 2012. PMID: 22731815

4

A new, sensitive ecto-5'-nucleotidase assay for compound screening.

Freundlieb M, Zimmermann H, Müller CE. Freundlieb M, et al. Among authors: zimmermann h. Anal Biochem. 2014 Feb 1;446:53-8. doi: 10.1016/j.ab.2013.10.012. Epub 2013 Oct 19. Anal Biochem. 2014. PMID: 24144488

5

Polyoxometalates--potent and selective ecto-nucleotidase inhibitors.

Lee SY, Fiene A, Li W, Hanck T, Brylev KA, Fedorov VE, Lecka J, Haider A, Pietzsch HJ, Zimmermann H, Sévigny J, Kortz U, Stephan H, Müller CE. Lee SY, et al. Among authors: zimmermann h. Biochem Pharmacol. 2015 Jan 15;93(2):171-81. doi: 10.1016/j.bcp.2014.11.002. Epub 2014 Nov 13. Biochem Pharmacol. 2015. PMID: 25449596

6

α,β-Methylene-ADP (AOPCP) Derivatives and Analogues: Development of Potent and Selective ecto-5'-Nucleotidase (CD73) Inhibitors.

Bhattarai S, Freundlieb M, Pippel J, Meyer A, Abdelrahman A, Fiene A, Lee SY, Zimmermann H, Yegutkin GG, Sträter N, El-Tayeb A, Müller CE. Bhattarai S, et al. Among authors: zimmermann h. J Med Chem. 2015 Aug 13;58(15):6248-63. doi: 10.1021/acs.jmedchem.5b00802. Epub 2015 Jul 30. J Med Chem. 2015. PMID: 26147331

7

Structure-Activity Relationship of Purine and Pyrimidine Nucleotides as Ecto-5'-Nucleotidase (CD73) Inhibitors.

Junker A, Renn C, Dobelmann C, Namasivayam V, Jain S, Losenkova K, Irjala H, Duca S, Balasubramanian R, Chakraborty S, Börgel F, Zimmermann H, Yegutkin GG, Müller CE, Jacobson KA. Junker A, et al. Among authors: zimmermann h. J Med Chem. 2019 Apr 11;62(7):3677-3695. doi: 10.1021/acs.jmedchem.9b00164. Epub 2019 Mar 21. J Med Chem. 2019. PMID: 30895781 Free PMC article.

8

2-Substituted α,β-Methylene-ADP Derivatives: Potent Competitive Ecto-5'-nucleotidase (CD73) Inhibitors with Variable Binding Modes.

Bhattarai S, Pippel J, Scaletti E, Idris R, Freundlieb M, Rolshoven G, Renn C, Lee SY, Abdelrahman A, Zimmermann H, El-Tayeb A, Müller CE, Sträter N. Bhattarai S, et al. Among authors: zimmermann h. J Med Chem. 2020 Mar 26;63(6):2941-2957. doi: 10.1021/acs.jmedchem.9b01611. Epub 2020 Feb 28. J Med Chem. 2020. PMID: 32045236

9

Polyoxometalates--a new class of potent ecto-nucleoside triphosphate diphosphohydrolase (NTPDase) inhibitors.

Müller CE, Iqbal J, Baqi Y, Zimmermann H, Röllich A, Stephan H. Müller CE, et al. Among authors: zimmermann h. Bioorg Med Chem Lett. 2006 Dec 1;16(23):5943-7. doi: 10.1016/j.bmcl.2006.09.003. Epub 2006 Sep 25. Bioorg Med Chem Lett. 2006. PMID: 16997558

10

Capillary electrophoresis-based nanoscale assays for monitoring ecto-5'-nucleotidase activity and inhibition in preparations of recombinant enzyme and melanoma cell membranes.

Iqbal J, Jirovsky D, Lee SY, Zimmermann H, Müller CE. Iqbal J, et al. Among authors: zimmermann h. Anal Biochem. 2008 Feb 1;373(1):129-40. doi: 10.1016/j.ab.2007.09.028. Epub 2007 Sep 29. Anal Biochem. 2008. PMID: 17980347

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

1,544 results

Search Page