Klotz KN - Search Results

1

Synthesis and pharmacological characterization of a new series of 5,7-disubstituted-[1,2,4]triazolo[1,5-a][1,3,5]triazine derivatives as adenosine receptor antagonists: A preliminary inspection of ligand-receptor recognition process.

Pastorin G, Federico S, Paoletta S, Corradino M, Cateni F, Cacciari B, Klotz KN, Gao ZG, Jacobson KA, Spalluto G, Moro S. Pastorin G, et al. Among authors: klotz kn. Bioorg Med Chem. 2010 Apr 1;18(7):2524-36. doi: 10.1016/j.bmc.2010.02.039. Epub 2010 Feb 25. Bioorg Med Chem. 2010. PMID: 20304654 Free PMC article.

2

Adenosine receptor agonists: synthesis and biological evaluation of 1-deaza analogues of adenosine derivatives.

Cristalli G, Franchetti P, Grifantini M, Vittori S, Klotz KN, Lohse MJ. Cristalli G, et al. Among authors: klotz kn. J Med Chem. 1988 Jun;31(6):1179-83. doi: 10.1021/jm00401a018. J Med Chem. 1988. PMID: 3373486

3

Synthesis of new delta 2-isoxazoline derivatives and their pharmacological characterization as beta-adrenergic receptor antagonists.

Conti P, Dallanoce C, De Amici M, De Micheli C, Klotz KN. Conti P, et al. Among authors: klotz kn. Bioorg Med Chem. 1998 Apr;6(4):401-8. doi: 10.1016/s0968-0896(97)10051-7. Bioorg Med Chem. 1998. PMID: 9597184

4

New substituted 9-alkylpurines as adenosine receptor ligands.

Camaioni E, Costanzi S, Vittori S, Volpini R, Klotz KN, Cristalli G. Camaioni E, et al. Among authors: klotz kn. Bioorg Med Chem. 1998 May;6(5):523-33. doi: 10.1016/s0968-0896(98)00007-8. Bioorg Med Chem. 1998. PMID: 9629466

5

8-(Sulfostyryl)xanthines: water-soluble A2A-selective adenosine receptor antagonists.

Müller CE, Sandoval-Ramírez J, Schobert U, Geis U, Frobenius W, Klotz KN. Müller CE, et al. Among authors: klotz kn. Bioorg Med Chem. 1998 Jun;6(6):707-19. doi: 10.1016/s0968-0896(98)00025-x. Bioorg Med Chem. 1998. PMID: 9681137

6

Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists.

Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Klotz KN, Leung E, Varani K, Gessi S, Merighi S, Borea PA. Baraldi PG, et al. Among authors: klotz kn. J Med Chem. 1999 Nov 4;42(22):4473-8. doi: 10.1021/jm991114s. J Med Chem. 1999. PMID: 10579811 No abstract available.

7

Water-soluble phosphate prodrugs of 1-propargyl-8-styrylxanthine derivatives, A(2A)-selective adenosine receptor antagonists.

Sauer R, Maurinsh J, Reith U, Fülle F, Klotz KN, Müller CE. Sauer R, et al. Among authors: klotz kn. J Med Chem. 2000 Feb 10;43(3):440-8. doi: 10.1021/jm9911480. J Med Chem. 2000. PMID: 10669571

8

Activation of the A3 adenosine receptor affects cell cycle progression and cell growth.

Brambilla R, Cattabeni F, Ceruti S, Barbieri D, Franceschi C, Kim YC, Jacobson KA, Klotz KN, Lohse MJ, Abbracchio MP. Brambilla R, et al. Among authors: klotz kn. Naunyn Schmiedebergs Arch Pharmacol. 2000 Mar;361(3):225-34. doi: 10.1007/s002109900186. Naunyn Schmiedebergs Arch Pharmacol. 2000. PMID: 10731034 Free PMC article.

9

[(3)H]MRE 3008F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors.

Varani K, Merighi S, Gessi S, Klotz KN, Leung E, Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Borea PA. Varani K, et al. Among authors: klotz kn. Mol Pharmacol. 2000 May;57(5):968-75. Mol Pharmacol. 2000. PMID: 10779381

10

7-Deazaadenines bearing polar substituents: structure-activity relationships of new A(1) and A(3) adenosine receptor antagonists.

Hess S, Müller CE, Frobenius W, Reith U, Klotz KN, Eger K. Hess S, et al. Among authors: klotz kn. J Med Chem. 2000 Nov 30;43(24):4636-46. doi: 10.1021/jm000967d. J Med Chem. 2000. PMID: 11101355

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