Structure-based design of potent and selective cell-permeable inhibitors of human beta-secretase (BACE-1).
Stachel SJ, Coburn CA, Steele TG, Jones KG, Loutzenhiser EF, Gregro AR, Rajapakse HA, Lai MT, Crouthamel MC, Xu M, Tugusheva K, Lineberger JE, Pietrak BL, Espeseth AS, Shi XP, Chen-Dodson E, Holloway MK, Munshi S, Simon AJ, Kuo L, Vacca JP.
Stachel SJ, et al. Among authors: munshi s.
J Med Chem. 2004 Dec 16;47(26):6447-50. doi: 10.1021/jm049379g.
J Med Chem. 2004.
PMID: 15588077