Costa G - Search Results

1

New structure-activity relationships of A- and D-ring modified steroidal aromatase inhibitors: design, synthesis, and biochemical evaluation.

Varela C, Tavares da Silva EJ, Amaral C, Correia da Silva G, Baptista T, Alcaro S, Costa G, Carvalho RA, Teixeira NA, Roleira FM. Varela C, et al. Among authors: costa g. J Med Chem. 2012 Apr 26;55(8):3992-4002. doi: 10.1021/jm300262w. Epub 2012 Apr 18. J Med Chem. 2012. PMID: 22475216

2

Synthesis of new 3-aryl-4,5-dihydropyrazole-1-carbothioamide derivatives. An investigation on their ability to inhibit monoamine oxidase.

Maccioni E, Alcaro S, Orallo F, Cardia MC, Distinto S, Costa G, Yanez M, Sanna ML, Vigo S, Meleddu R, Secci D. Maccioni E, et al. Among authors: costa g. Eur J Med Chem. 2010 Oct;45(10):4490-8. doi: 10.1016/j.ejmech.2010.07.009. Epub 2010 Jul 17. Eur J Med Chem. 2010. PMID: 20702005

3

3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: a new scaffold for the selective inhibition of monoamine oxidase B.

Maccioni E, Alcaro S, Cirilli R, Vigo S, Cardia MC, Sanna ML, Meleddu R, Yanez M, Costa G, Casu L, Matyus P, Distinto S. Maccioni E, et al. Among authors: costa g. J Med Chem. 2011 Sep 22;54(18):6394-8. doi: 10.1021/jm2002876. Epub 2011 Aug 17. J Med Chem. 2011. PMID: 21777011

4

GRID-based three-dimensional pharmacophores II: PharmBench, a benchmark data set for evaluating pharmacophore elucidation methods.

Cross S, Ortuso F, Baroni M, Costa G, Distinto S, Moraca F, Alcaro S, Cruciani G. Cross S, et al. Among authors: costa g. J Chem Inf Model. 2012 Oct 22;52(10):2599-608. doi: 10.1021/ci300154n. Epub 2012 Sep 21. J Chem Inf Model. 2012. PMID: 22970854

5

Identification and characterization of new DNA G-quadruplex binders selected by a combination of ligand and structure-based virtual screening approaches.

Alcaro S, Musetti C, Distinto S, Casatti M, Zagotto G, Artese A, Parrotta L, Moraca F, Costa G, Ortuso F, Maccioni E, Sissi C. Alcaro S, et al. Among authors: costa g. J Med Chem. 2013 Feb 14;56(3):843-55. doi: 10.1021/jm3013486. Epub 2013 Jan 22. J Med Chem. 2013. PMID: 23294188

6

Toward the design of new DNA G-quadruplex ligands through rational analysis of polymorphism and binding data.

Artese A, Costa G, Distinto S, Moraca F, Ortuso F, Parrotta L, Alcaro S. Artese A, et al. Among authors: costa g. Eur J Med Chem. 2013 Oct;68:139-49. doi: 10.1016/j.ejmech.2013.07.022. Epub 2013 Aug 11. Eur J Med Chem. 2013. PMID: 23974014

7

Identification of new natural DNA G-quadruplex binders selected by a structure-based virtual screening approach.

Artese A, Costa G, Ortuso F, Parrotta L, Alcaro S. Artese A, et al. Among authors: costa g. Molecules. 2013 Sep 30;18(10):12051-70. doi: 10.3390/molecules181012051. Molecules. 2013. PMID: 24084014 Free PMC article.

8

New insights into the biological properties of Crocus sativus L.: chemical modifications, human monoamine oxidases inhibition and molecular modeling studies.

De Monte C, Carradori S, Chimenti P, Secci D, Mannina L, Alcaro F, Petzer A, N'Da CI, Gidaro MC, Costa G, Alcaro S, Petzer JP. De Monte C, et al. Among authors: costa g. Eur J Med Chem. 2014 Jul 23;82:164-71. doi: 10.1016/j.ejmech.2014.05.048. Epub 2014 May 22. Eur J Med Chem. 2014. PMID: 24904963

9

Bioactive compounds of Crocus sativus L. and their semi-synthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents.

De Monte C, Bizzarri B, Gidaro MC, Carradori S, Mollica A, Luisi G, Granese A, Alcaro S, Costa G, Basilico N, Parapini S, Scaltrito MM, Masia C, Sisto F. De Monte C, et al. Among authors: costa g. J Enzyme Inhib Med Chem. 2015 Dec;30(6):1027-33. doi: 10.3109/14756366.2014.1001755. Epub 2015 Sep 4. J Enzyme Inhib Med Chem. 2015. PMID: 25766747 Free article.

10

(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies.

D'Ascenzio M, Chimenti P, Gidaro MC, De Monte C, De Vita D, Granese A, Scipione L, Di Santo R, Costa G, Alcaro S, Yáñez M, Carradori S. D'Ascenzio M, et al. Among authors: costa g. J Enzyme Inhib Med Chem. 2015 Dec;30(6):908-19. doi: 10.3109/14756366.2014.987138. Epub 2015 Sep 25. J Enzyme Inhib Med Chem. 2015. PMID: 25807300

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