Garabadzhiu AV - Search Results

1

The 26S proteasome is a multifaceted target for anti-cancer therapies.

Grigoreva TA, Tribulovich VG, Garabadzhiu AV, Melino G, Barlev NA. Grigoreva TA, et al. Among authors: garabadzhiu av. Oncotarget. 2015 Sep 22;6(28):24733-49. doi: 10.18632/oncotarget.4619. Oncotarget. 2015. PMID: 26295307 Free PMC article. Review.

2

Proapoptotic modification of substituted isoindolinones as MDM2-p53 inhibitors.

Grigoreva TA, Novikova DS, Petukhov AV, Gureev MA, Garabadzhiu AV, Melino G, Barlev NA, Tribulovich VG. Grigoreva TA, et al. Among authors: garabadzhiu av. Bioorg Med Chem Lett. 2017 Dec 1;27(23):5197-5202. doi: 10.1016/j.bmcl.2017.10.049. Epub 2017 Oct 20. Bioorg Med Chem Lett. 2017. PMID: 29089230

3

Amino acids as chiral derivatizing agents for antiproliferative substituted N-benzyl isoindolinones.

Grigoreva TA, Novikova DS, Gureev MA, Garabadzhiu AV, Tribulovich VG. Grigoreva TA, et al. Among authors: garabadzhiu av. Chirality. 2018 Jun;30(6):785-797. doi: 10.1002/chir.22854. Epub 2018 Mar 25. Chirality. 2018. PMID: 29575058

4

Simulation of MDM2 N-terminal domain conformational lability in the presence of imidazoline based inhibitors of MDM2-p53 protein-protein interaction.

Gureev M, Novikova D, Grigoreva T, Vorona S, Garabadzhiu A, Tribulovich V. Gureev M, et al. J Comput Aided Mol Des. 2020 Jan;34(1):55-70. doi: 10.1007/s10822-019-00260-6. Epub 2019 Nov 28. J Comput Aided Mol Des. 2020. PMID: 31781989

5

Advanced palladium free approach to the synthesis of substituted alkene oxindoles via aluminum-promoted Knoevenagel reaction.

Novikova DS, Grigoreva TA, Zolotarev AA, Garabadzhiu AV, Tribulovich VG. Novikova DS, et al. Among authors: garabadzhiu av. RSC Adv. 2018 Oct 10;8(60):34543-34551. doi: 10.1039/c8ra07576j. eCollection 2018 Oct 4. RSC Adv. 2018. PMID: 35548634 Free PMC article.

6

Design, in silico prioritization and biological profiling of apoptosis-inducing lactams amenable by the Castagnoli-Cushman reaction.

Krasavin M, Gureyev MA, Dar'in D, Bakulina O, Chizhova M, Lepikhina A, Novikova D, Grigoreva T, Ivanov G, Zhumagalieva A, Garabadzhiu AV, Tribulovich VG. Krasavin M, et al. Among authors: garabadzhiu av. Bioorg Med Chem. 2018 May 15;26(9):2651-2673. doi: 10.1016/j.bmc.2018.04.036. Epub 2018 Apr 18. Bioorg Med Chem. 2018. PMID: 29691156

7

Inhibition of Neutrophil Elastase and Cathepsin G As a New Approach to the Treatment of Psoriasis: From Fundamental Biology to Development of New Target-Specific Drugs.

Krasavin MY, Gureev MA, Garabadzhiu AV, Pashkin AY, Zhukov AS, Khairutdinov VR, Samtsov AV, Shvets VI. Krasavin MY, et al. Among authors: garabadzhiu av. Dokl Biochem Biophys. 2019 Jul;487(1):272-276. doi: 10.1134/S1607672919040082. Epub 2019 Sep 26. Dokl Biochem Biophys. 2019. PMID: 31559596

8

Preclinical efficacy investigation of human neutrophil elastase inhibitor sivelestat in animal model of psoriasis.

Zhukov AS, Khairutdinov VR, Samtsov AV, Krasavin M, Garabadzhiu AV. Zhukov AS, et al. Among authors: garabadzhiu av. Skin Health Dis. 2021 Dec 30;2(2):e90. doi: 10.1002/ski2.90. eCollection 2022 Jun. Skin Health Dis. 2021. PMID: 35677925 Free PMC article.

9

Identification of small-molecule elastase inhibitors as antagonists of IL-36 cytokine activation.

Sullivan GP, Davidovich PB, Sura-Trueba S, Belotcerkovskaya E, Henry CM, Clancy DM, Zinoveva A, Mametnabiev T, Garabadzhiu AV, Martin SJ. Sullivan GP, et al. Among authors: garabadzhiu av. FEBS Open Bio. 2018 Mar 25;8(5):751-763. doi: 10.1002/2211-5463.12406. eCollection 2018 May. FEBS Open Bio. 2018. PMID: 29744290 Free PMC article.

10

Suppressing IL-36-driven inflammation using peptide pseudosubstrates for neutrophil proteases.

Sullivan GP, Henry CM, Clancy DM, Mametnabiev T, Belotcerkovskaya E, Davidovich P, Sura-Trueba S, Garabadzhiu AV, Martin SJ. Sullivan GP, et al. Among authors: garabadzhiu av. Cell Death Dis. 2018 Mar 7;9(3):378. doi: 10.1038/s41419-018-0385-4. Cell Death Dis. 2018. PMID: 29515113 Free PMC article. Clinical Trial.

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