Discovery, synthesis and mechanism study of 2,3,5-substituted [1,2,4]-thiadiazoles as covalent inhibitors targeting 3C-Like protease of SARS-CoV-2.
Ren P, Yu C, Zhang R, Nie T, Hu Q, Li H, Zhang X, Zhang X, Li S, Liu L, Dai W, Li J, Xu Y, Su H, Zhang L, Liu H, Bai F.
Ren P, et al. Among authors: liu h, liu l.
Eur J Med Chem. 2023 Mar 5;249:115129. doi: 10.1016/j.ejmech.2023.115129. Epub 2023 Jan 18.
Eur J Med Chem. 2023.
PMID: 36702052
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