Georg GI - Search Results

1

BET Bromodomain Inhibitors with One-Step Synthesis Discovered from Virtual Screen.

Ayoub AM, Hawk LML, Herzig RJ, Jiang J, Wisniewski AJ, Gee CT, Zhao P, Zhu JY, Berndt N, Offei-Addo NK, Scott TG, Qi J, Bradner JE, Ward TR, Schönbrunn E, Georg GI, Pomerantz WCK. Ayoub AM, et al. Among authors: georg gi. J Med Chem. 2017 Jun 22;60(12):4805-4817. doi: 10.1021/acs.jmedchem.6b01336. Epub 2017 Jun 7. J Med Chem. 2017. PMID: 28535045 Free PMC article.

2

Butitaxel analogues: synthesis and structure-activity relationships.

Ali SM, Hoemann MZ, Aubé J, Georg GI, Mitscher LA, Jayasinghe LR. Ali SM, et al. Among authors: georg gi. J Med Chem. 1997 Jan 17;40(2):236-41. doi: 10.1021/jm960505t. J Med Chem. 1997. PMID: 9003522

3

A one-step synthesis of a deuterated paclitaxel analogue: 10-deacetoxy-(10alpha-2H)paclitaxel.

Dutta D, Hadd H, Vander Velde DG, Georg GI. Dutta D, et al. Among authors: georg gi. Bioorg Med Chem Lett. 1999 Dec 6;9(23):3277-8. doi: 10.1016/s0960-894x(99)00609-5. Bioorg Med Chem Lett. 1999. PMID: 10612584

4

Total synthesis and antitubulin activity of c10 analogues of cryptophycin-24.

Buck SB, Huff JK, Himes RH, Georg GI. Buck SB, et al. Among authors: georg gi. J Med Chem. 2004 Jan 29;47(3):696-702. doi: 10.1021/jm030278c. J Med Chem. 2004. PMID: 14736249

5

Total synthesis and anti-tubulin activity of epi-c3 analogues of cryptophycin-24.

Buck SB, Huff JK, Himes RH, Georg GI. Buck SB, et al. Among authors: georg gi. J Med Chem. 2004 Jul 1;47(14):3697-9. doi: 10.1021/jm030555f. J Med Chem. 2004. PMID: 15214797

6

Design, synthesis, and antiproliferative and CDK2-cyclin a inhibitory activity of novel flavopiridol analogues.

Ahn YM, Vogeti L, Liu CJ, Santhapuram HK, White JM, Vasandani V, Mitscher LA, Lushington GH, Hanson PR, Powell DR, Himes RH, Roby KF, Ye Q, Georg GI. Ahn YM, et al. Among authors: georg gi. Bioorg Med Chem. 2007 Jan 15;15(2):702-13. doi: 10.1016/j.bmc.2006.10.063. Epub 2006 Nov 1. Bioorg Med Chem. 2007. PMID: 17123821 Free PMC article.

7

Synthesis, in vitro and in vivo cytotoxicity of 6,7-diaryl-2,3,8,8a-tetrahydroindolizin-5(1H)-ones.

Kimball FS, Tunoori AR, Victory SF, Dutta D, White JM, Himes RH, Georg GI. Kimball FS, et al. Among authors: georg gi. Bioorg Med Chem Lett. 2007 Aug 15;17(16):4703-7. doi: 10.1016/j.bmcl.2007.05.103. Epub 2007 Jun 13. Bioorg Med Chem Lett. 2007. PMID: 17614274 Free PMC article.

8

Synthesis of a quinolone library from ynones.

Ward TR, Turunen BJ, Haack T, Neuenswander B, Shadrick W, Georg GI. Ward TR, et al. Among authors: georg gi. Tetrahedron Lett. 2009 Nov 25;50(47):6494-9497. doi: 10.1016/j.tetlet.2009.09.024. Tetrahedron Lett. 2009. PMID: 20161410 Free PMC article.

9

Discovery of a potential allosteric ligand binding site in CDK2.

Betzi S, Alam R, Martin M, Lubbers DJ, Han H, Jakkaraj SR, Georg GI, Schönbrunn E. Betzi S, et al. Among authors: georg gi. ACS Chem Biol. 2011 May 20;6(5):492-501. doi: 10.1021/cb100410m. Epub 2011 Feb 22. ACS Chem Biol. 2011. PMID: 21291269 Free PMC article.

10

Synthesis and evaluation of eight- and four-membered iminosugar analogues as inhibitors of testicular ceramide-specific glucosyltransferase, testicular β-glucosidase 2, and other glycosidases.

Lee JC, Francis S, Dutta D, Gupta V, Yang Y, Zhu JY, Tash JS, Schönbrunn E, Georg GI. Lee JC, et al. Among authors: georg gi. J Org Chem. 2012 Apr 6;77(7):3082-98. doi: 10.1021/jo202054g. Epub 2012 Mar 20. J Org Chem. 2012. PMID: 22432895 Free PMC article.

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