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Identification of an imidazopyridine scaffold to generate potent and selective TYK2 inhibitors that demonstrate activity in an in vivo psoriasis model.
Bioorg Med Chem Lett. 2017 Sep 15;27(18):4370-4376. doi: 10.1016/j.bmcl.2017.08.022. Epub 2017 Aug 12.
Bioorg Med Chem Lett. 2017.
PMID: 28830649
Lead optimization of a 4-aminopyridine benzamide scaffold to identify potent, selective, and orally bioavailable TYK2 inhibitors.
Liang J, van Abbema A, Balazs M, Barrett K, Berezhkovsky L, Blair W, Chang C, Delarosa D, DeVoss J, Driscoll J, Eigenbrot C, Ghilardi N, Gibbons P, Halladay J, Johnson A, Kohli PB, Lai Y, Liu Y, Lyssikatos J, Mantik P, Menghrajani K, Murray J, Peng I, Sambrone A, Shia S, Shin Y, Smith J, Sohn S, Tsui V, Ultsch M, Wu LC, Xiao Y, Yang W, Young J, Zhang B, Zhu BY, Magnuson S.
Liang J, et al. Among authors: mantik p.
J Med Chem. 2013 Jun 13;56(11):4521-36. doi: 10.1021/jm400266t. Epub 2013 May 29.
J Med Chem. 2013.
PMID: 23668484
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Lead identification of novel and selective TYK2 inhibitors.
Liang J, Tsui V, Van Abbema A, Bao L, Barrett K, Beresini M, Berezhkovskiy L, Blair WS, Chang C, Driscoll J, Eigenbrot C, Ghilardi N, Gibbons P, Halladay J, Johnson A, Kohli PB, Lai Y, Liimatta M, Mantik P, Menghrajani K, Murray J, Sambrone A, Xiao Y, Shia S, Shin Y, Smith J, Sohn S, Stanley M, Ultsch M, Zhang B, Wu LC, Magnuson S.
Liang J, et al. Among authors: mantik p.
Eur J Med Chem. 2013 Sep;67:175-87. doi: 10.1016/j.ejmech.2013.03.070. Epub 2013 May 14.
Eur J Med Chem. 2013.
PMID: 23867602
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Cyclodextrin Reduces Intravenous Toxicity of a Model Compound.
Mantik P, Xie M, Wong H, La H, Steigerwalt RW, Devanaboyina U, Ganem G, Shih D, Flygare JA, Fairbrother WJ, Chakravarty P, Russell D, Fernandez GE, Narang AS.
Mantik P, et al.
J Pharm Sci. 2019 Jun;108(6):1934-1943. doi: 10.1016/j.xphs.2019.01.004. Epub 2019 Jan 11.
J Pharm Sci. 2019.
PMID: 30639736
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Probing the Protein-Excipient Interaction in the Orally Delivered Protein by Solid-State Hydrogen-Deuterium Exchange Mass Spectrometry and Molecular Dynamics.
Pan X, Lenka S, Davis J, Nagapudi K, Mantik P, Saggu M, Dai L, Cadang L, Zhang HM, Zhang J, Izadi S, Yang F, Wei B.
Pan X, et al. Among authors: mantik p.
Anal Chem. 2024 Jan 16;96(2):802-809. doi: 10.1021/acs.analchem.3c04255. Epub 2023 Dec 28.
Anal Chem. 2024.
PMID: 38155586
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Predicting Long-Term Stability of an Oral Delivered Antibody Drug Product with Accelerated Stability Assessment Program Modeling.
Dai L, Davis J, Nagapudi K, Mantik P, Zhang K, Pellett JD, Wei B.
Dai L, et al. Among authors: mantik p.
Mol Pharm. 2024 Jan 1;21(1):325-332. doi: 10.1021/acs.molpharmaceut.3c00877. Epub 2023 Dec 7.
Mol Pharm. 2024.
PMID: 38060811
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