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DNA intercalators based on (1,10-phenanthrolin-2-yl)isoxazolidin-5-yl core with better growth inhibition and selectivity than cisplatin upon head and neck squamous cells carcinoma.
Eur J Med Chem. 2018 Jan 1;143:583-590. doi: 10.1016/j.ejmech.2017.11.067. Epub 2017 Nov 26.
Eur J Med Chem. 2018.
PMID: 29207341
Novel isoxazole polycyclic aromatic hydrocarbons as DNA-intercalating agents.
Rescifina A, Varrica MG, Carnovale C, Romeo G, Chiacchio U.
Rescifina A, et al. Among authors: varrica mg.
Eur J Med Chem. 2012 May;51:163-73. doi: 10.1016/j.ejmech.2012.02.038. Epub 2012 Feb 25.
Eur J Med Chem. 2012.
PMID: 22405647
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Recent advances in small organic molecules as DNA intercalating agents: synthesis, activity, and modeling.
Rescifina A, Zagni C, Varrica MG, Pistarà V, Corsaro A.
Rescifina A, et al. Among authors: varrica mg.
Eur J Med Chem. 2014 Mar 3;74:95-115. doi: 10.1016/j.ejmech.2013.11.029. Epub 2014 Jan 3.
Eur J Med Chem. 2014.
PMID: 24448420
Review.
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