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Identification of the Binding Site of Apical Membrane Antigen 1 (AMA1) Inhibitors Using a Paramagnetic Probe.
ChemMedChem. 2019 Mar 5;14(5):603-612. doi: 10.1002/cmdc.201800802. Epub 2019 Feb 13.
ChemMedChem. 2019.
PMID: 30653832
Ligand-induced conformational change of Plasmodium falciparum AMA1 detected using 19F NMR.
Ge X, MacRaild CA, Devine SM, Debono CO, Wang G, Scammells PJ, Scanlon MJ, Anders RF, Foley M, Norton RS.
Ge X, et al. Among authors: debono co.
J Med Chem. 2014 Aug 14;57(15):6419-27. doi: 10.1021/jm500390g. Epub 2014 Aug 5.
J Med Chem. 2014.
PMID: 25068708
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Structure and dynamics of apical membrane antigen 1 from Plasmodium falciparum FVO.
Lim SS, Yang W, Krishnarjuna B, Kannan Sivaraman K, Chandrashekaran IR, Kass I, MacRaild CA, Devine SM, Debono CO, Anders RF, Scanlon MJ, Scammells PJ, Norton RS, McGowan S.
Lim SS, et al. Among authors: debono co.
Biochemistry. 2014 Nov 25;53(46):7310-20. doi: 10.1021/bi5012089. Epub 2014 Nov 14.
Biochemistry. 2014.
PMID: 25360546
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Solution NMR characterization of apical membrane antigen 1 and small molecule interactions as a basis for designing new antimalarials.
Krishnarjuna B, Lim SS, Devine SM, Debono CO, Lam R, Chandrashekaran IR, Jaipuria G, Yagi H, Atreya HS, Scanlon MJ, MacRaild CA, Scammells PJ, Norton RS.
Krishnarjuna B, et al. Among authors: debono co.
J Mol Recognit. 2016 Jun;29(6):281-91. doi: 10.1002/jmr.2529. Epub 2016 Jan 24.
J Mol Recognit. 2016.
PMID: 26804042
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Promiscuous 2-aminothiazoles (PrATs): a frequent hitting scaffold.
Devine SM, Mulcair MD, Debono CO, Leung EW, Nissink JW, Lim SS, Chandrashekaran IR, Vazirani M, Mohanty B, Simpson JS, Baell JB, Scammells PJ, Norton RS, Scanlon MJ.
Devine SM, et al. Among authors: debono co.
J Med Chem. 2015 Feb 12;58(3):1205-14. doi: 10.1021/jm501402x. Epub 2015 Jan 16.
J Med Chem. 2015.
PMID: 25559643
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