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Design of Potent and Selective Covalent Inhibitors of Bruton's Tyrosine Kinase Targeting an Inactive Conformation.
ACS Med Chem Lett. 2019 Sep 6;10(10):1467-1472. doi: 10.1021/acsmedchemlett.9b00317. eCollection 2019 Oct 10.
ACS Med Chem Lett. 2019.
PMID: 31620235
Free PMC article.
Discovery of LOU064 (Remibrutinib), a Potent and Highly Selective Covalent Inhibitor of Bruton's Tyrosine Kinase.
Angst D, Gessier F, Janser P, Vulpetti A, Wälchli R, Beerli C, Littlewood-Evans A, Dawson J, Nuesslein-Hildesheim B, Wieczorek G, Gutmann S, Scheufler C, Hinniger A, Zimmerlin A, Funhoff EG, Pulz R, Cenni B.
Angst D, et al. Among authors: pulz r.
J Med Chem. 2020 May 28;63(10):5102-5118. doi: 10.1021/acs.jmedchem.9b01916. Epub 2020 Mar 4.
J Med Chem. 2020.
PMID: 32083858
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Design and Synthesis of Inhibitors of the E3 Ligase SMAD Specific E3 Ubiquitin Protein Ligase 1 as a Treatment for Lung Remodeling in Pulmonary Arterial Hypertension.
Shaw DE, Smith N, Beerli R, Cotesta S, D'Alessandro PL, Edwards AM, Lattmann R, Lizos D, Pulz R, Rooney L, Sohal B, Rynn C, Taylor J, Troxler T, Williams G, Guth S, Rowlands D.
Shaw DE, et al. Among authors: pulz r.
J Med Chem. 2023 Jun 22;66(12):8130-8139. doi: 10.1021/acs.jmedchem.3c00229. Epub 2023 Jun 9.
J Med Chem. 2023.
PMID: 37294287
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Leydig cell number and sperm production decrease induced by chronic ametryn exposure: a negative impact on animal reproductive health.
Dantas TA, Cancian G, Neodini DN, Mano DR, Capucho C, Predes FS, Pulz RB, Pigoso AA, Dolder H, Severi-Aguiar GD.
Dantas TA, et al. Among authors: pulz rb.
Environ Sci Pollut Res Int. 2015 Jun;22(11):8526-35. doi: 10.1007/s11356-014-4010-5. Epub 2015 Jan 6.
Environ Sci Pollut Res Int. 2015.
PMID: 25561257
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New polyhydroxylated pyrrolidines derived from enantiopure 3,6-dihydro-2H-1,2-oxazines.
Pulz R, Al-Harrasi A, Reissig HU.
Pulz R, et al.
Org Lett. 2002 Jul 11;4(14):2353-5. doi: 10.1021/ol0260573.
Org Lett. 2002.
PMID: 12098245
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