Tuccinardi T - Search Results

1

1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors.

D'Ascenzio M, Secci D, Carradori S, Zara S, Guglielmi P, Cirilli R, Pierini M, Poli G, Tuccinardi T, Angeli A, Supuran CT. D'Ascenzio M, et al. Among authors: tuccinardi t. J Med Chem. 2020 Mar 12;63(5):2470-2488. doi: 10.1021/acs.jmedchem.9b01434. Epub 2020 Feb 4. J Med Chem. 2020. PMID: 31972093

2

Study on affinity profile toward native human and bovine adenosine receptors of a series of 1,8-naphthyridine derivatives.

Ferrarini PL, Betti L, Cavallini T, Giannaccini G, Lucacchini A, Manera C, Martinelli A, Ortore G, Saccomanni G, Tuccinardi T. Ferrarini PL, et al. Among authors: tuccinardi t. J Med Chem. 2004 Jun 3;47(12):3019-31. doi: 10.1021/jm030977p. J Med Chem. 2004. PMID: 15163184

3

Amber force field implementation, molecular modelling study, synthesis and MMP-1/MMP-2 inhibition profile of (R)- and (S)-N-hydroxy-2-(N-isopropoxybiphenyl-4-ylsulfonamido)-3-methylbutanamides.

Tuccinardi T, Martinelli A, Nuti E, Carelli P, Balzano F, Uccello-Barretta G, Murphy G, Rossello A. Tuccinardi T, et al. Bioorg Med Chem. 2006 Jun 15;14(12):4260-76. doi: 10.1016/j.bmc.2006.01.056. Epub 2006 Feb 17. Bioorg Med Chem. 2006. PMID: 16483784

4

Pharmacophore based receptor modeling: the case of adenosine A3 receptor antagonists. An approach to the optimization of protein models.

Tafi A, Bernardini C, Botta M, Corelli F, Andreini M, Martinelli A, Ortore G, Baraldi PG, Fruttarolo F, Borea PA, Tuccinardi T. Tafi A, et al. Among authors: tuccinardi t. J Med Chem. 2006 Jul 13;49(14):4085-97. doi: 10.1021/jm051112+. J Med Chem. 2006. PMID: 16821770

5

Synthesis of anthranylaldoxime derivatives as estrogen receptor ligands and computational prediction of binding modes.

Tuccinardi T, Bertini S, Martinelli A, Minutolo F, Ortore G, Placanica G, Prota G, Rapposelli S, Carlson KE, Katzenellenbogen JA, Macchia M. Tuccinardi T, et al. J Med Chem. 2006 Aug 10;49(16):5001-12. doi: 10.1021/jm060560u. J Med Chem. 2006. PMID: 16884312

6

Analysis of human carbonic anhydrase II: docking reliability and receptor-based 3D-QSAR study.

Tuccinardi T, Nuti E, Ortore G, Supuran CT, Rossello A, Martinelli A. Tuccinardi T, et al. J Chem Inf Model. 2007 Mar-Apr;47(2):515-25. doi: 10.1021/ci600469w. Epub 2007 Feb 13. J Chem Inf Model. 2007. PMID: 17295464

7

5-amino-2-phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one: a versatile scaffold to obtain potent and selective A3 adenosine receptor antagonists.

Da Settimo F, Primofiore G, Taliani S, Marini AM, La Motta C, Simorini F, Salerno S, Sergianni V, Tuccinardi T, Martinelli A, Cosimelli B, Greco G, Novellino E, Ciampi O, Trincavelli ML, Martini C. Da Settimo F, et al. Among authors: tuccinardi t. J Med Chem. 2007 Nov 15;50(23):5676-84. doi: 10.1021/jm0708376. Epub 2007 Oct 10. J Med Chem. 2007. PMID: 17927167

8

New 1,8-naphthyridine and quinoline derivatives as CB2 selective agonists.

Manera C, Cascio MG, Benetti V, Allarà M, Tuccinardi T, Martinelli A, Saccomanni G, Vivoli E, Ghelardini C, Di Marzo V, Ferrarini PL. Manera C, et al. Among authors: tuccinardi t. Bioorg Med Chem Lett. 2007 Dec 1;17(23):6505-10. doi: 10.1016/j.bmcl.2007.09.089. Epub 2007 Oct 1. Bioorg Med Chem Lett. 2007. PMID: 17942307

9

Homology modeling and receptor-based 3D-QSAR study of carbonic anhydrase IX.

Tuccinardi T, Ortore G, Rossello A, Supuran CT, Martinelli A. Tuccinardi T, et al. J Chem Inf Model. 2007 Nov-Dec;47(6):2253-62. doi: 10.1021/ci700214j. Epub 2007 Oct 20. J Chem Inf Model. 2007. PMID: 17949069

10

Dual inhibitors of matrix metalloproteinases and carbonic anhydrases: iminodiacetyl-based hydroxamate-benzenesulfonamide conjugates.

Marques SM, Nuti E, Rossello A, Supuran CT, Tuccinardi T, Martinelli A, Santos MA. Marques SM, et al. Among authors: tuccinardi t. J Med Chem. 2008 Dec 25;51(24):7968-79. doi: 10.1021/jm800964f. J Med Chem. 2008. PMID: 19053764

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